Compile Data Set for Download or QSAR
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Found 5 Enz. Inhib. hit(s) with all data for entry = 5547
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Dumlupinar University

LigandPNGBDBM87064(Sulfonamide derivative, 5)
Affinity DataKi:  4.20E+3nM IC50:  2.53E+3nMAssay Description:The enzyme activities in the absence of drugs or chemicals were taken as 100%. For each drug or chemical, an activity%-(drug) graph was drawn and dr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione-disulfide reductase(Escherichia coli)
Dumlupinar University

LigandPNGBDBM87062(Sulfonamide derivative, 2)
Affinity DataKi:  6.10E+3nM IC50:  4.50E+3nMAssay Description:The enzyme activities in the absence of drugs or chemicals were taken as 100%. For each drug or chemical, an activity%-(drug) graph was drawn and dr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlutathione-disulfide reductase(Escherichia coli)
Dumlupinar University

LigandPNGBDBM87061(Sulfonamide derivative, 1)
Affinity DataKi:  7.23E+4nM IC50:  4.71E+4nMAssay Description:The enzyme activities in the absence of drugs or chemicals were taken as 100%. For each drug or chemical, an activity%-(drug) graph was drawn and dr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Dumlupinar University

LigandPNGBDBM87063(Sulfonamide derivative, 3)
Affinity DataKi:  8.78E+4nM IC50:  6.01E+4nMAssay Description:The enzyme activities in the absence of drugs or chemicals were taken as 100%. For each drug or chemical, an activity%-(drug) graph was drawn and dr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target6-phosphogluconate dehydrogenase, decarboxylating(Homo sapiens (Human))
Dumlupinar University

LigandPNGBDBM50043906(CHEMBL269001 | Dorzolamide | MK-507 | US10172837, ...)
Affinity DataKi:  3.14E+6nM IC50:  1.41E+6nMAssay Description:The enzyme activities in the absence of drugs or chemicals were taken as 100%. For each drug or chemical, an activity%-(drug) graph was drawn and dr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed