Compile Data Set for Download or QSAR
maximum 50k data
Found 68 Enz. Inhib. hit(s) with all data for entry = 50026587
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263219(3-(5-cyano-4-(4-methyl-1H-indol-5-ylamino)thieno[2...)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263265(3-(5-cyano-4-(4-methyl-1H-indol-5-ylamino)thieno[2...)
Affinity DataIC50:  2nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50262606(3-methyl-4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-...)
Affinity DataIC50:  3.5nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263218(3-(5-cyano-4-(4-methyl-1H-indol-5-ylamino)thieno[2...)
Affinity DataIC50:  12nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263266(3-(5-cyano-4-(4-methyl-1H-indol-5-ylamino)thieno[2...)
Affinity DataIC50:  15nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50262605(4-(4-methyl-1H-indol-5-ylamino)-2-(3-(pyrrolidin-1...)
Affinity DataIC50:  22nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50:  25nMAssay Description:Inhibition of FYNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase HCK(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50:  26nMAssay Description:Inhibition of HCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50:  28nMAssay Description:Inhibition of LYNMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263133(2-(3-(3-hydroxypyrrolidin-1-yl)-3-oxoprop-1-enyl)-...)
Affinity DataIC50:  41nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263217(4-(4-methyl-1H-indol-5-ylamino)-2-(3-(4-methylpipe...)
Affinity DataIC50:  43nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50:  46nMAssay Description:Inhibition of LCKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263268(3-(5-cyano-4-(4-methyl-1H-indol-5-ylamino)thieno[2...)
Affinity DataIC50:  48nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263175(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(piperi...)
Affinity DataIC50:  48nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263176(4-(4-methyl-1H-indol-5-ylamino)-2-(3-morpholino-3-...)
Affinity DataIC50:  53nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50262604(4-(4-methyl-1H-indol-5-ylamino)-2-(3-(pyrrolidine-...)
Affinity DataIC50:  58nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263218(3-(5-cyano-4-(4-methyl-1H-indol-5-ylamino)thieno[2...)
Affinity DataIC50:  67nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263217(4-(4-methyl-1H-indol-5-ylamino)-2-(3-(4-methylpipe...)
Affinity DataIC50:  73nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263216(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pipera...)
Affinity DataIC50:  88nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263301(3-(5-cyano-4-(4-methyl-1H-indol-5-ylamino)thieno[2...)
Affinity DataIC50:  100nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50262605(4-(4-methyl-1H-indol-5-ylamino)-2-(3-(pyrrolidin-1...)
Affinity DataIC50:  100nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263267(3-(5-cyano-4-(4-methyl-1H-indol-5-ylamino)thieno[2...)
Affinity DataIC50:  110nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50262607(4-(1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrolidin-1-yl...)
Affinity DataIC50:  130nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263300(3-(5-cyano-4-(4-methyl-1H-indol-5-ylamino)thieno[2...)
Affinity DataIC50:  150nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263174((S)-2-(3-(3-(dimethylamino)pyrrolidin-1-yl)-3-oxop...)
Affinity DataIC50:  170nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263173((R)-2-(3-(3-(dimethylamino)pyrrolidin-1-yl)-3-oxop...)
Affinity DataIC50:  180nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50262604(4-(4-methyl-1H-indol-5-ylamino)-2-(3-(pyrrolidine-...)
Affinity DataIC50:  180nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263216(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pipera...)
Affinity DataIC50:  200nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263265(3-(5-cyano-4-(4-methyl-1H-indol-5-ylamino)thieno[2...)
Affinity DataIC50:  250nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263303(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50:  250nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50:  330nMAssay Description:Inhibition of SRCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263302(3-(5-cyano-4-(4-methyl-1H-indol-5-ylamino)thieno[2...)
Affinity DataIC50:  330nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263174((S)-2-(3-(3-(dimethylamino)pyrrolidin-1-yl)-3-oxop...)
Affinity DataIC50:  340nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263302(3-(5-cyano-4-(4-methyl-1H-indol-5-ylamino)thieno[2...)
Affinity DataIC50:  370nMAssay Description:Inhibition of PKCthetaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50262606(3-methyl-4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-...)
Affinity DataIC50:  380nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263301(3-(5-cyano-4-(4-methyl-1H-indol-5-ylamino)thieno[2...)
Affinity DataIC50:  420nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263173((R)-2-(3-(3-(dimethylamino)pyrrolidin-1-yl)-3-oxop...)
Affinity DataIC50:  430nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263175(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(piperi...)
Affinity DataIC50:  450nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263133(2-(3-(3-hydroxypyrrolidin-1-yl)-3-oxoprop-1-enyl)-...)
Affinity DataIC50:  450nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263266(3-(5-cyano-4-(4-methyl-1H-indol-5-ylamino)thieno[2...)
Affinity DataIC50:  500nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263267(3-(5-cyano-4-(4-methyl-1H-indol-5-ylamino)thieno[2...)
Affinity DataIC50:  500nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263300(3-(5-cyano-4-(4-methyl-1H-indol-5-ylamino)thieno[2...)
Affinity DataIC50:  790nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263268(3-(5-cyano-4-(4-methyl-1H-indol-5-ylamino)thieno[2...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263303(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263219(3-(5-cyano-4-(4-methyl-1H-indol-5-ylamino)thieno[2...)
Affinity DataIC50:  2.10E+3nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C epsilon type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of PKCepsilonMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C delta type(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263176(4-(4-methyl-1H-indol-5-ylamino)-2-(3-morpholino-3-...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of PKCdeltaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ITK/TSK(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50263132(4-(4-methyl-1H-indol-5-ylamino)-2-(3-oxo-3-(pyrrol...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of ITKMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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