Compile Data Set for Download or QSAR
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Found 25 Enz. Inhib. hit(s) with all data for entry = 50038636
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM27659(1-(3-{[(2S)-2-aminopropanamido]methyl}phenyl)-N-be...)
Affinity DataIC50:  80nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262871(2-{3-[((S)-2-Amino-propionylamino)-methyl]-phenyl}...)
Affinity DataIC50:  160nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262920(1-(3-(((S)-2-aminopropanamido)methyl)phenyl)-N-((R...)
Affinity DataIC50:  180nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262826(1-(3-((2-aminoacetamido)methyl)phenyl)-N-(3-(methy...)
Affinity DataIC50:  230nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262985(CHEMBL478195 | benzyl 1-(3-(((S)-2-aminopropanamid...)
Affinity DataIC50:  600nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262921(1-(3-(((S)-2-aminopropanamido)methyl)phenyl)-N-phe...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262876(1-(3-(((S)-2-aminopropanamido)methyl)phenyl)-N-phe...)
Affinity DataIC50:  1.32E+3nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262869(2-{3-[(2-Amino-acetylamino)-methyl]-phenyl}-5-trif...)
Affinity DataIC50:  1.42E+3nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262982(2-{3-[(2-Amino-acetylamino)-methyl]-phenyl}-5-trif...)
Affinity DataIC50:  1.80E+3nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262877(1-(3-(((S)-2-aminopropanamido)methyl)phenyl)-N-ben...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262922(1-(3-(((S)-2-aminopropanamido)methyl)phenyl)-N-cyc...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262919(1-(3-(((S)-2-aminopropanamido)methyl)phenyl)-N-((S...)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262825(1-(3-((2-aminoacetamido)methyl)phenyl)-N-phenyl-3-...)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262823(1-(3-((2-aminoacetamido)methyl)phenyl)-N-methyl-3-...)
Affinity DataIC50:  1.06E+4nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262870(2-{3-[(3-Amino-propionylamino)-methyl]-phenyl}-5-t...)
Affinity DataIC50:  1.69E+4nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262872(2-{3-[((R)-2-Amino-propionylamino)-methyl]-phenyl}...)
Affinity DataIC50:  2.01E+4nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 3 [N508S](Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM27659(1-(3-{[(2S)-2-aminopropanamido]methyl}phenyl)-N-be...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of GST-tagged PRMT3 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein arginine N-methyltransferase 1 [11-371](Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM27659(1-(3-{[(2S)-2-aminopropanamido]methyl}phenyl)-N-be...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of GST-tagged PRMT1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262824(1-(3-((2-aminoacetamido)methyl)phenyl)-N,N-dimethy...)
Affinity DataIC50:  2.98E+4nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262874(2-{3-[(2-Amino-3,3,3-trifluoro-propionylamino)-met...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262875(2-{3-[(2-Methylamino-acetylamino)-methyl]-phenyl}-...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262873(2-{3-[(2-Amino-2-methyl-propionylamino)-methyl]-ph...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262983((S)-1-(4-((2-aminopropanamido)methyl)phenyl)-N-ben...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50377950(CHEMBL1162995)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-arginine methyltransferase CARM1(Homo sapiens (Human))
Bristol-Myers Squibb Pharmaceutical Research And Development

Curated by ChEMBL
LigandPNGBDBM50262984(1-(2-(((S)-2-aminopropanamido)methyl)phenyl)-N-ben...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human GST-tagged CARM1 by methylation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed