Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glucocorticoid (RAT) | BDBM39347![]() (CLOBETASOL PROPIONATE | MLS000028708 | SMR00005874...) | PDB UniProtKB/SwissProt GoogleScholar | Purchase CHEBI DrugBank PC cid PC sid UniChem Patents Similars | Article PubMed | n/a | n/a | 3.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Mitsubishi Kasei Corporation Curated by ChEMBL | Assay Description Competitive displacement of [3H]dexamethasone from glucocorticoid receptor of rat liver cytosol | J Med Chem 34: 2468-73 (1991) Article DOI: 10.1021/jm00112a023 BindingDB Entry DOI: 10.7270/Q2W096H9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid (RAT) | BDBM50009401![]() (CHEMBL315931 | Succinic acid 17-(2-chloro-acetyl)-...) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.20 | n/a | n/a | n/a | n/a | n/a | n/a |
Mitsubishi Kasei Corporation Curated by ChEMBL | Assay Description Competitive displacement of [3H]dexamethasone from glucocorticoid receptor of rat liver cytosol | J Med Chem 34: 2468-73 (1991) Article DOI: 10.1021/jm00112a023 BindingDB Entry DOI: 10.7270/Q2W096H9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid (RAT) | BDBM50421892![]() (Alphatrex | BETAMETHASONE DIPROPIONATE | Diprolene...) | PDB UniProtKB/SwissProt GoogleScholar | Purchase CHEBI PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 5.30 | n/a | n/a | n/a | n/a | n/a | n/a |
Mitsubishi Kasei Corporation Curated by ChEMBL | Assay Description Competitive displacement of [3H]dexamethasone from glucocorticoid receptor of rat liver cytosol | J Med Chem 34: 2468-73 (1991) Article DOI: 10.1021/jm00112a023 BindingDB Entry DOI: 10.7270/Q2W096H9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid (RAT) | BDBM50009403![]() (CHEMBL81387 | Pentanedioic acid 17-(2-chloro-acety...) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 9.70 | n/a | n/a | n/a | n/a | n/a | n/a |
Mitsubishi Kasei Corporation Curated by ChEMBL | Assay Description Competitive displacement of [3H]dexamethasone from glucocorticoid receptor of rat liver cytosol | J Med Chem 34: 2468-73 (1991) Article DOI: 10.1021/jm00112a023 BindingDB Entry DOI: 10.7270/Q2W096H9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid (RAT) | BDBM50009402![]() (CHEMBL83845 | Succinic acid tert-butyl ester 17-(2...) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 11 | n/a | n/a | n/a | n/a | n/a | n/a |
Mitsubishi Kasei Corporation Curated by ChEMBL | Assay Description Competitive displacement of [3H]dexamethasone from glucocorticoid receptor of rat liver cytosol | J Med Chem 34: 2468-73 (1991) Article DOI: 10.1021/jm00112a023 BindingDB Entry DOI: 10.7270/Q2W096H9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid (RAT) | BDBM50009406![]() (CHEMBL311802 | Succinic acid 17-(2-chloro-acetyl)-...) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | 12 | n/a | n/a | n/a | n/a | n/a | n/a |
Mitsubishi Kasei Corporation Curated by ChEMBL | Assay Description Competitive displacement of [3H]dexamethasone from glucocorticoid receptor of rat liver cytosol | J Med Chem 34: 2468-73 (1991) Article DOI: 10.1021/jm00112a023 BindingDB Entry DOI: 10.7270/Q2W096H9 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glucocorticoid (RAT) | BDBM50009405![]() (CHEMBL311457 | Succinic acid mono-[17-(2-chloro-ac...) | PDB UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | n/a | n/a | >150 | n/a | n/a | n/a | n/a | n/a | n/a |
Mitsubishi Kasei Corporation Curated by ChEMBL | Assay Description Competitive displacement of [3H]dexamethasone from glucocorticoid receptor of rat liver cytosol | J Med Chem 34: 2468-73 (1991) Article DOI: 10.1021/jm00112a023 BindingDB Entry DOI: 10.7270/Q2W096H9 | |||||||||||
More data for this Ligand-Target Pair |