Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50009591![]() (1-(2-Methyl-1-phenyl-cyclohexyl)-piperidine | CHEM...) | PDB Reactome pathway UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 11 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Istituto Superiore di Sanità Curated by ChEMBL | Assay Description Binding affinity by displacement of [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate preparation of rat brain without ce... | J Med Chem 34: 2615-23 (1991) Article DOI: 10.1021/jm00112a041 BindingDB Entry DOI: 10.7270/Q22806K3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50009591![]() (1-(2-Methyl-1-phenyl-cyclohexyl)-piperidine | CHEM...) | PDB Reactome pathway UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 25 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Istituto Superiore di Sanità Curated by ChEMBL | Assay Description Binding affinity by displacement of [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate preparation of rat brain without ce... | J Med Chem 34: 2615-23 (1991) Article DOI: 10.1021/jm00112a041 BindingDB Entry DOI: 10.7270/Q22806K3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM83449![]() (1-(1-phenylcyclohexyl)piperidine;hydrochloride | M...) | PDB Reactome pathway UniProtKB/SwissProt GoogleScholar | Purchase DrugBank KEGG PC cid PC sid PDB UniChem Similars | Article PubMed | 53 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Istituto Superiore di Sanità Curated by ChEMBL | Assay Description Binding affinity of the compound was determined by displacement of [3H]-TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate pre... | J Med Chem 34: 2615-23 (1991) Article DOI: 10.1021/jm00112a041 BindingDB Entry DOI: 10.7270/Q22806K3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50009591![]() (1-(2-Methyl-1-phenyl-cyclohexyl)-piperidine | CHEM...) | PDB Reactome pathway UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 100 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Istituto Superiore di Sanità Curated by ChEMBL | Assay Description Binding affinity of the compound was determined by displacement of [3H]-TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate pre... | J Med Chem 34: 2615-23 (1991) Article DOI: 10.1021/jm00112a041 BindingDB Entry DOI: 10.7270/Q22806K3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50009592![]() (CHEMBL424610 | cis-1-(4-Methyl-1-phenyl-cyclohexyl...) | PDB Reactome pathway UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 166 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Istituto Superiore di Sanità Curated by ChEMBL | Assay Description Binding affinity of the compound was determined by displacement of [3H]-TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate pre... | J Med Chem 34: 2615-23 (1991) Article DOI: 10.1021/jm00112a041 BindingDB Entry DOI: 10.7270/Q22806K3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50009592![]() (CHEMBL424610 | cis-1-(4-Methyl-1-phenyl-cyclohexyl...) | PDB Reactome pathway UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Patents Similars | Article PubMed | 617 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Istituto Superiore di Sanità Curated by ChEMBL | Assay Description Binding affinity of the compound was determined by displacement of [3H]-TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate pre... | J Med Chem 34: 2615-23 (1991) Article DOI: 10.1021/jm00112a041 BindingDB Entry DOI: 10.7270/Q22806K3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50009591![]() (1-(2-Methyl-1-phenyl-cyclohexyl)-piperidine | CHEM...) | PDB Reactome pathway UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.18E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Istituto Superiore di Sanità Curated by ChEMBL | Assay Description Binding affinity of the compound was determined by displacement of [3H]-TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate pre... | J Med Chem 34: 2615-23 (1991) Article DOI: 10.1021/jm00112a041 BindingDB Entry DOI: 10.7270/Q22806K3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50009591![]() (1-(2-Methyl-1-phenyl-cyclohexyl)-piperidine | CHEM...) | PDB Reactome pathway UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.94E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Istituto Superiore di Sanità Curated by ChEMBL | Assay Description Binding affinity by displacement of [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate preparation of rat brain without ce... | J Med Chem 34: 2615-23 (1991) Article DOI: 10.1021/jm00112a041 BindingDB Entry DOI: 10.7270/Q22806K3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50009590![]() (CHEMBL86824 | cis-C-(2-Methyl-1-piperidin-1-yl-cyc...) | PDB Reactome pathway UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.70E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Istituto Superiore di Sanità Curated by ChEMBL | Assay Description Binding affinity of the compound was determined by displacement of [3H]-TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate pre... | J Med Chem 34: 2615-23 (1991) Article DOI: 10.1021/jm00112a041 BindingDB Entry DOI: 10.7270/Q22806K3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50009591![]() (1-(2-Methyl-1-phenyl-cyclohexyl)-piperidine | CHEM...) | PDB Reactome pathway UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 7.40E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Istituto Superiore di Sanità Curated by ChEMBL | Assay Description Binding affinity by displacement of [3H]TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate preparation of rat brain without ce... | J Med Chem 34: 2615-23 (1991) Article DOI: 10.1021/jm00112a041 BindingDB Entry DOI: 10.7270/Q22806K3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50009590![]() (CHEMBL86824 | cis-C-(2-Methyl-1-piperidin-1-yl-cyc...) | PDB Reactome pathway UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Istituto Superiore di Sanità Curated by ChEMBL | Assay Description Binding affinity of the compound was determined by displacement of [3H]-TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate pre... | J Med Chem 34: 2615-23 (1991) Article DOI: 10.1021/jm00112a041 BindingDB Entry DOI: 10.7270/Q22806K3 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Glutamate receptor ionotropic, NMDA 1 (RAT) | BDBM50009593![]() (C-Phenyl-C-(1-piperidin-1-yl-cyclohexyl)-methylene...) | PDB Reactome pathway UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 3.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Istituto Superiore di Sanità Curated by ChEMBL | Assay Description Binding affinity of the compound was determined by displacement of [3H]-TCP from PCP N-methyl-D-aspartate glutamate receptor of tissue homogenate pre... | J Med Chem 34: 2615-23 (1991) Article DOI: 10.1021/jm00112a041 BindingDB Entry DOI: 10.7270/Q22806K3 | |||||||||||
More data for this Ligand-Target Pair |