Compile Data Set for Download or QSAR
maximum 50k data
Found 58 Enz. Inhib. hit(s) with all data for entry = 50027634
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275059((Z)-1-(Benzo[b]thiophen-3-ylmethylene)-6-methyl-4-...)
Affinity DataIC50:  970nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275013((Z)-1-((1H-Indol-2-yl)methylene)-6-methyl-4-thioxo...)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50274962((Z)-1-((5-Methoxybenzofuran-2-yl)methylene)-6-meth...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275239((Z)-6-Methyl-1-((5-methylfuran-2-yl)methylene)-4-t...)
Affinity DataIC50:  2.70E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50274964((Z)-1-((7-Methoxybenzofuran-2-yl)methylene)-6-meth...)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275015((Z)-1-((6-Methoxy-1H-indol-2-yl)methylene)-6-methy...)
Affinity DataIC50:  3.10E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275274((Z)-6-Methyl-1-((5-phenylthiophen-2-yl)methylene)-...)
Affinity DataIC50:  3.40E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275060((Z)-1-[(4-Methoxy-1-benzothien-3-yl)methylene]-6-m...)
Affinity DataIC50:  3.80E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275241((Z)-6-Methyl-1-((5-phenylfuran-2-yl)methylene)-4-t...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275134((Z)-1-((1H-Indol-7-yl)methylene)-6-methyl-4-thioxo...)
Affinity DataIC50:  4.10E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275098((Z)-6-Methyl-1-((1-methyl-1H-indol-3-yl)methylene)...)
Affinity DataIC50:  4.30E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275240((Z)-1-(Furan-2-ylmethylene)-6-methyl-4-thioxo-4,5-...)
Affinity DataIC50:  4.40E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50274991((Z)-1-(Benzo[b]thiophen-2-ylmethylene)-6-methylfur...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275014((Z)-1-((5-Methoxy-1H-indol-2-yl)methylene)-6-methy...)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275094((Z)-1-((6-Methoxybenzo[b]thiophen-3-yl)methylene)-...)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50274829((Z)-6-Methyl-1-((5-phenylthiophen-2-yl)methylene)f...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50274987((Z)-1-((6-(Benzyloxy)-5-methoxybenzofuran-2-yl)met...)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275093((Z)-1-((5-Methoxybenzo[b]thiophen-3-yl)methylene)-...)
Affinity DataIC50:  5.10E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50274990((Z)-1-((6-Methoxybenzo[b]thiophen-2-yl)methylene)-...)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275017((Z)-1-((5-Fluoro-6-methoxy-1H-indol-3-yl)methylene...)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50274961((Z)-1-((4-Methoxybenzofuran-2-yl)methylene)-6-meth...)
Affinity DataIC50:  6.70E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50274963((Z)-1-((6-Methoxybenzofuran-2-yl)methylene)-6-meth...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275273((Z)-6-Methyl-1-((5-methylthiophen-2-yl)methylene)-...)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275095((Z)-1-((5-Bromobenzo[b]thiophen-3-yl)methylene)-6-...)
Affinity DataIC50:  7.50E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50274960((Z)-1-(Benzofuran-2-ylmethylene)-6-methyl-4-thioxo...)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275096((Z)-1-(Benzo[b]thiophen-3-ylmethylene)-6-methylfur...)
Affinity DataIC50:  8.50E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275242((Z)-6-Methyl-1-(thiophen-2-ylmethylene)-4-thioxo-4...)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50274988((Z)-1-(Benzo[b]thiophen-2-ylmethylene)-6-methyl-4-...)
Affinity DataIC50:  9.50E+3nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50274989((Z)-1-((5-Methoxybenzo[b]thiophen-2-yl)methylene)-...)
Affinity DataIC50:  1.31E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275133((Z)-1-(Benzo[b]thiophen-3-ylmethylene)-6-methyl-4-...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275132((Z)-6-Methyl-1-((1-methyl-1H-indol-3-yl)methylene)...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275097((Z)-1-((1H-Indol-3-yl)methylene)-6-methyl-4-thioxo...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50274830((Z)-1-((1H-Pyrrol-2-yl)methylene)-6-methylfuro[3,4...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50274828((Z)-6-Methyl-1-((5-methylfuran-2-yl)methylene)furo...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50274827((Z)-1-(Biphenyl-4-ylmethylene)-6-methyl-4-thioxo-4...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50274826((Z)-N-(4-((6-Methyl-3-oxo-4-thioxo-4,5-dihydrofuro...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50274825((Z)-1-(4-(Dimethylamino)benzylidene)-6-methyl-4-th...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275318((Z)-6-Methyl-1-(4-(methylthio)benzylidene)-4-thiox...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275317((Z)-6-Methyl-4-thioxo-1-(4-(trifluoromethoxy)benzy...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275316((Z)-1-(4-Methoxybenzylidene)-6-methyl-4-thioxo-4,5...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275315((Z)-6-Methyl-4-thioxo-1-(4-(trifluoromethyl)benzyl...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275314((Z)-6-Methyl-1-(4-methylbenzylidene)-4-thioxo-4,5-...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275313((Z)-1-(4-Chlorobenzylidene)-6-methyl-4-thioxo-4,5-...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275279((Z)-1-(4-Fluorobenzylidene)-6-methyl-4-thioxo-4,5-...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275278((Z)-1-Benzylidene-6-methyl-4-thioxo-4,5-dihydrofur...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275277((Z)-6-Methyl-1-((1-methyl-1H-pyrrol-2-yl)methylene...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275276((Z)-1-((1H-Imidazol-2-yl)methylene)-6-methyl-4-thi...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275275((Z)-1-((1H-Pyrrol-2-yl)methylene)-6-methyl-4-thiox...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275058((Z)-1-(Benzofuran-3-ylmethylene)-6-methyl-4-thioxo...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPerforin-1(Homo sapiens (Human))
University Of Auckland

Curated by ChEMBL
LigandPNGBDBM50275057((Z)-6-Methyl-1-((1-methyl-1H-indol-2-yl)methylene)...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of recombinant perforin (unknown origin)-mediated lysis of human Jurkat T cells by 51Cr release assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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