Compile Data Set for Download or QSAR
maximum 50k data
Found 44 Enz. Inhib. hit(s) with all data for entry = 3101
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28020(6-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-2-(2,6-di...)
Affinity DataIC50:  60nMAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27985(2-{[(3-chlorophenyl)methyl]amino}-N-(2-phenoxyethy...)
Affinity DataIC50:  70nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28017(6-{[(2S)-1-hydroxy-3-phenylpropan-2-yl]amino}-N-(2...)
Affinity DataIC50:  76nMAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28019(6-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-(2-phen...)
Affinity DataIC50:  130nMAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28018(2-(2,6-dimethoxypyridin-3-yl)-6-{[(2S)-1-hydroxy-3...)
Affinity DataIC50:  140nMAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27998(2-{[(2S)-1-hydroxy-3-phenylpropan-2-yl]amino}-N-(2...)
Affinity DataIC50:  150nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28014(2-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-[1-(4-c...)
Affinity DataIC50:  150nMAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27988(2-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-N-(2-phen...)
Affinity DataIC50:  150nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28015(6-[benzyl(ethyl)amino]-N-(2-phenoxyethyl)-2-(3,4,5...)
Affinity DataIC50:  154nMAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28021(6-{[(3-chlorophenyl)methyl]amino}-N-(2-phenoxyethy...)
Affinity DataIC50:  162nMAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28022(6-{[(3-chlorophenyl)methyl]amino}-2-(2,6-dimethoxy...)
Affinity DataIC50:  197nMAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27979(2-[benzyl(ethyl)amino]-N-(2-phenoxyethyl)-4-(3,4,5...)
Affinity DataIC50:  200nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28012(2-[(2H-1,3-benzodioxol-5-ylmethyl)amino]-4-(2,6-di...)
Affinity DataIC50:  220nMAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27993(2-{[2-(2-methoxyphenyl)ethyl]amino}-N-(2-phenoxyet...)
Affinity DataIC50:  340nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27987(2-{[(3-methoxyphenyl)methyl]amino}-N-(2-phenoxyeth...)
Affinity DataIC50:  340nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28013(N-(2H-1,3-benzodioxol-5-ylmethyl)-4-(2,6-dimethoxy...)
Affinity DataIC50:  360nMAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28011(2-[benzyl(ethyl)amino]-4-(2,6-dimethoxypyridin-3-y...)
Affinity DataIC50:  360nMAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27991(N-(2-phenoxyethyl)-2-[(2-phenylethyl)amino]-4-(3,4...)
Affinity DataIC50:  400nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27982(2-[benzyl(methyl)amino]-N-(2-phenoxyethyl)-4-(3,4,...)
Affinity DataIC50:  470nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27981(2-(benzylamino)-N-(2-phenoxyethyl)-4-(3,4,5-trimet...)
Affinity DataIC50:  730nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27994(2-{[2-(3-methoxyphenyl)ethyl]amino}-N-(2-phenoxyet...)
Affinity DataIC50:  1.00E+3nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28016(6-[benzyl(ethyl)amino]-2-(2,6-dimethoxypyridin-3-y...)
Affinity DataIC50:  1.05E+3nMAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27992(2-[methyl(2-phenylethyl)amino]-N-(2-phenoxyethyl)-...)
Affinity DataIC50:  1.50E+3nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28004(2-[benzyl(ethyl)amino]-N-(4-phenylbutyl)-4-(3,4,5-...)
Affinity DataIC50:  1.80E+3nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28003(2-[benzyl(ethyl)amino]-N-(3-phenylpropyl)-4-(3,4,5...)
Affinity DataIC50:  2.10E+3nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27980(2-[(3-methylbutyl)amino]-N-(2-phenoxyethyl)-4-(3,4...)
Affinity DataIC50:  2.20E+3nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27995(2-{[2-(4-methoxyphenyl)ethyl]amino}-N-(2-phenoxyet...)
Affinity DataIC50:  2.80E+3nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27986(2-{[(4-methoxyphenyl)methyl]amino}-N-(2-phenoxyeth...)
Affinity DataIC50:  3.10E+3nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27983(2-{[(2-chlorophenyl)methyl]amino}-N-(2-phenoxyethy...)
Affinity DataIC50:  4.90E+3nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28009(2-[benzyl(methyl)amino]-4-(3,4-dimethoxyphenyl)-N-...)
Affinity DataIC50:  6.90E+3nMAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27984(2-{[(2-methylphenyl)methyl]amino}-N-(2-phenoxyethy...)
Affinity DataIC50:  1.00E+4nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28008(2-[benzyl(methyl)amino]-N-(2-phenoxyethyl)-4-[4-(t...)
Affinity DataIC50:  1.89E+4nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27999(2-{[(2R)-1-hydroxy-3-phenylpropan-2-yl]amino}-N-(2...)
Affinity DataIC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27997(N-(2-phenoxyethyl)-2-{[2-(pyridin-3-yl)ethyl]amino...)
Affinity DataIC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27996(N-(2-phenoxyethyl)-2-{[2-(pyridin-2-yl)ethyl]amino...)
Affinity DataIC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27990(N-(2-phenoxyethyl)-2-[(pyridin-3-ylmethyl)amino]-4...)
Affinity DataIC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM27989(N-(2-phenoxyethyl)-2-[(pyridin-2-ylmethyl)amino]-4...)
Affinity DataIC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28000(2-[benzyl(ethyl)amino]-N-(2-phenoxyethyl)-4-phenyl...)
Affinity DataIC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28001(2-[benzyl(ethyl)amino]-4-cyclohexyl-N-(2-phenoxyet...)
Affinity DataIC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28010(2-[benzyl(methyl)amino]-4-(3,5-dimethoxyphenyl)-N-...)
Affinity DataIC50: >3.00E+4nMAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28007(2-[benzyl(methyl)amino]-4-(4-methoxyphenyl)-N-(2-p...)
Affinity DataIC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28002(2-[benzyl(ethyl)amino]-N-(2-phenylethyl)-4-(3,4,5-...)
Affinity DataIC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28005(2-[benzyl(methyl)amino]-4-(2-methoxyphenyl)-N-(2-p...)
Affinity DataIC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetExtracellular calcium-sensing receptor(Homo sapiens (Human))
Bristol-Myers Squibb

LigandPNGBDBM28006(2-[benzyl(methyl)amino]-4-(3-methoxyphenyl)-N-(2-p...)
Affinity DataIC50: >3.00E+4nMpH: 7.5 T: 2°CAssay Description:Antagonist activity of test compounds was measured in HEK293 cells stably expressing the human recombinant CaR (HEK-CaR) by determining the ability o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed