Compile Data Set for Download or QSAR
maximum 50k data
Found 63 Enz. Inhib. hit(s) with all data for entry = 50028496
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50196246(2-(1-(3-(6-benzoyl-1-propylnaphthalen-2-yloxy)prop...)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257255(2-{1-[3-(6-Benzyl-1-propyl-naphthalen-2-yloxy)-pro...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257300(2-{1-[3-(6-Acetyl-1-propyl-naphthalen-2-yloxy)-pro...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257301(2-Methyl-2-(1-{3-[1-propyl-6-(pyridine-4-carbonyl)...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257302(2-(1-{3-[6-(Furan-3-carbonyl)-1-propyl-naphthalen-...)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257303(2-(1-{3-[6-(4-Fluoro-benzoyl)-1-propyl-naphthalen-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257304(2-(1-{3-[6-(4-Methoxy-benzoyl)-1-propyl-naphthalen...)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257305(2-Methyl-2-(1-{3-[4-(naphthalene-2-carbonyl)-2-pro...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257306(2-Methyl-2-(1-{3-[4-(naphthalene-2-carbonyl)-2-pro...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257307(2-(1-{3-[4-(Biphenyl-4-carbonyl)-2-propyl-phenoxy]...)
Affinity DataEC50:  1.92E+3nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257308(2-(1-{3-[4-(Biphenyl-4-carbonyl)-2-propyl-phenoxy]...)
Affinity DataEC50:  4.07E+3nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257309(2-{1-[3-(4-Benzoyl-2-propyl-phenoxy)-propyl]-1H-in...)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257358(2-{1-[3-(4-Benzoyl-2-propyl-phenoxy)-propyl]-1H-in...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257359(2-(1-{3-[4-(4-Fluoro-benzoyl)-2-propyl-phenoxy]-pr...)
Affinity DataEC50:  130nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257360(2-(1-{3-[4-(4-Methoxy-benzoyl)-2-propyl-phenoxy]-p...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257361(2-{1-[3-(6-Benzoyl-1-propyl-naphthalen-2-yloxy)-pr...)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257362(2-{1-[3-(6-Benzoyl-1-propyl-naphthalen-2-yloxy)-pr...)
Affinity DataEC50:  240nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257363(2-(1-{3-[4-(Biphenyl-4-carbonyl)-2-propylphenoxy]p...)
Affinity DataEC50:  3.99E+3nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257364(2-(1-{3-[4-(Biphenyl-4-carbonyl)-2-propyl-phenoxy]...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARalpha receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50196246(2-(1-(3-(6-benzoyl-1-propylnaphthalen-2-yloxy)prop...)
Affinity DataEC50:  650nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257254(2-{1-[3-(5-Benzoyl-1-propyl-naphthalen-2-yloxy)-pr...)
Affinity DataEC50:  3.50E+3nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257255(2-{1-[3-(6-Benzyl-1-propyl-naphthalen-2-yloxy)-pro...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257300(2-{1-[3-(6-Acetyl-1-propyl-naphthalen-2-yloxy)-pro...)
Affinity DataEC50:  1.07E+3nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257301(2-Methyl-2-(1-{3-[1-propyl-6-(pyridine-4-carbonyl)...)
Affinity DataEC50:  2.07E+3nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257302(2-(1-{3-[6-(Furan-3-carbonyl)-1-propyl-naphthalen-...)
Affinity DataEC50:  430nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257303(2-(1-{3-[6-(4-Fluoro-benzoyl)-1-propyl-naphthalen-...)
Affinity DataEC50:  2.12E+3nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257304(2-(1-{3-[6-(4-Methoxy-benzoyl)-1-propyl-naphthalen...)
Affinity DataEC50:  510nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257305(2-Methyl-2-(1-{3-[4-(naphthalene-2-carbonyl)-2-pro...)
Affinity DataEC50:  370nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257306(2-Methyl-2-(1-{3-[4-(naphthalene-2-carbonyl)-2-pro...)
Affinity DataEC50:  2.80E+3nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257307(2-(1-{3-[4-(Biphenyl-4-carbonyl)-2-propyl-phenoxy]...)
Affinity DataEC50:  120nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257308(2-(1-{3-[4-(Biphenyl-4-carbonyl)-2-propyl-phenoxy]...)
Affinity DataEC50:  300nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257309(2-{1-[3-(4-Benzoyl-2-propyl-phenoxy)-propyl]-1H-in...)
Affinity DataEC50:  420nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257358(2-{1-[3-(4-Benzoyl-2-propyl-phenoxy)-propyl]-1H-in...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257359(2-(1-{3-[4-(4-Fluoro-benzoyl)-2-propyl-phenoxy]-pr...)
Affinity DataEC50:  900nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257360(2-(1-{3-[4-(4-Methoxy-benzoyl)-2-propyl-phenoxy]-p...)
Affinity DataEC50:  470nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257361(2-{1-[3-(6-Benzoyl-1-propyl-naphthalen-2-yloxy)-pr...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257362(2-{1-[3-(6-Benzoyl-1-propyl-naphthalen-2-yloxy)-pr...)
Affinity DataEC50:  540nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257363(2-(1-{3-[4-(Biphenyl-4-carbonyl)-2-propylphenoxy]p...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257364(2-(1-{3-[4-(Biphenyl-4-carbonyl)-2-propyl-phenoxy]...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM28681(5-[(4-{2-[methyl(pyridin-2-yl)amino]ethoxy}phenyl)...)
Affinity DataEC50:  220nMAssay Description:Agonist activity at human PPARgamma receptor by cell based transactivation assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50196246(2-(1-(3-(6-benzoyl-1-propylnaphthalen-2-yloxy)prop...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257254(2-{1-[3-(5-Benzoyl-1-propyl-naphthalen-2-yloxy)-pr...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257255(2-{1-[3-(6-Benzyl-1-propyl-naphthalen-2-yloxy)-pro...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257300(2-{1-[3-(6-Acetyl-1-propyl-naphthalen-2-yloxy)-pro...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257301(2-Methyl-2-(1-{3-[1-propyl-6-(pyridine-4-carbonyl)...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257302(2-(1-{3-[6-(Furan-3-carbonyl)-1-propyl-naphthalen-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257303(2-(1-{3-[6-(4-Fluoro-benzoyl)-1-propyl-naphthalen-...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50257304(2-(1-{3-[6-(4-Methoxy-benzoyl)-1-propyl-naphthalen...)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human PPARdelta receptor by cell based transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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