Compile Data Set for Download or QSAR
maximum 50k data
Found 52 Enz. Inhib. hit(s) with all data for entry = 50038829
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277789(3-(1H-tetrazol-5-yl)-5-(2,3,5-trifluorophenyl)-1,4...)
Affinity DataIC50:  70nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277789(3-(1H-tetrazol-5-yl)-5-(2,3,5-trifluorophenyl)-1,4...)
Affinity DataIC50:  70nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277790(5-(3,5-difluorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,...)
Affinity DataIC50:  70nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277790(5-(3,5-difluorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,...)
Affinity DataIC50:  70nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277789(3-(1H-tetrazol-5-yl)-5-(2,3,5-trifluorophenyl)-1,4...)
Affinity DataIC50:  80nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277789(3-(1H-tetrazol-5-yl)-5-(2,3,5-trifluorophenyl)-1,4...)
Affinity DataIC50:  80nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277788(5-(3-fluorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,6-te...)
Affinity DataIC50:  80nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277752(5-(2,3-difluorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,...)
Affinity DataIC50:  90nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277788(5-(3-fluorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,6-te...)
Affinity DataIC50:  140nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277752(5-(2,3-difluorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,...)
Affinity DataIC50:  140nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277787(5-(3-chlorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,6-te...)
Affinity DataIC50:  140nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM23515(CHEMBL573 | Niacin | Nicotinic Acid | [5, 6-3H]-ni...)
Affinity DataIC50:  140nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM23515(CHEMBL573 | Niacin | Nicotinic Acid | [5, 6-3H]-ni...)
Affinity DataIC50:  140nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277672(5-butyl-3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocyc...)
Affinity DataIC50:  210nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277672(5-butyl-3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocyc...)
Affinity DataIC50:  210nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277671(5-propyl-3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocy...)
Affinity DataIC50:  260nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277787(5-(3-chlorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,6-te...)
Affinity DataIC50:  290nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277710(5-phenyl-3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocy...)
Affinity DataIC50:  310nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277672(5-butyl-3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocyc...)
Affinity DataIC50:  340nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277672(5-butyl-3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocyc...)
Affinity DataIC50:  340nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277786(5-(2-fluorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,6-te...)
Affinity DataIC50:  340nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277786(5-(2-fluorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,6-te...)
Affinity DataIC50:  410nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277710(5-phenyl-3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocy...)
Affinity DataIC50:  430nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277751(5-(3,4-difluorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,...)
Affinity DataIC50:  520nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277751(5-(3,4-difluorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,...)
Affinity DataIC50:  610nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277671(5-propyl-3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocy...)
Affinity DataIC50:  690nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277749(5-(2,5-difluorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,...)
Affinity DataIC50:  760nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277707(5-hexyl-3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocyc...)
Affinity DataIC50:  800nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277749(5-(2,5-difluorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,...)
Affinity DataIC50:  850nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277707(5-hexyl-3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocyc...)
Affinity DataIC50:  870nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50273099(3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocyclopenta[...)
Affinity DataIC50:  1.20E+3nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277670(5-ethyl-3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocyc...)
Affinity DataIC50:  1.30E+3nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50273099(3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocyclopenta[...)
Affinity DataIC50:  1.50E+3nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277748(5-(2,4-difluorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,...)
Affinity DataIC50:  1.60E+3nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277747(5-(4-fluorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,6-te...)
Affinity DataIC50:  1.70E+3nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277750(5-(2-chlorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,6-te...)
Affinity DataIC50:  1.90E+3nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277748(5-(2,4-difluorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,...)
Affinity DataIC50:  2.40E+3nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277708(5-cyclopropyl-3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahy...)
Affinity DataIC50:  2.50E+3nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277709(5-cyclopentyl-3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahy...)
Affinity DataIC50:  2.50E+3nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277747(5-(4-fluorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,6-te...)
Affinity DataIC50:  2.70E+3nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277750(5-(2-chlorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,6-te...)
Affinity DataIC50:  3.10E+3nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277673(5-pentyl-3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocy...)
Affinity DataIC50:  3.60E+3nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277713(5-(4-chlorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,6-te...)
Affinity DataIC50:  4.00E+3nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277712(3-(1H-tetrazol-5-yl)-5-o-tolyl-1,4,5,6-tetrahydroc...)
Affinity DataIC50:  4.20E+3nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277670(5-ethyl-3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocyc...)
Affinity DataIC50:  4.60E+3nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277673(5-pentyl-3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahydrocy...)
Affinity DataIC50:  4.80E+3nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277713(5-(4-chlorophenyl)-3-(1H-tetrazol-5-yl)-1,4,5,6-te...)
Affinity DataIC50:  5.00E+3nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277708(5-cyclopropyl-3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahy...)
Affinity DataIC50:  5.20E+3nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277712(3-(1H-tetrazol-5-yl)-5-o-tolyl-1,4,5,6-tetrahydroc...)
Affinity DataIC50:  7.70E+3nMAssay Description:Displacement of [3H]nicotinic acid from human GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHydroxycarboxylic acid receptor 2(Mus musculus)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50277709(5-cyclopentyl-3-(1H-tetrazol-5-yl)-1,4,5,6-tetrahy...)
Affinity DataIC50:  9.00E+3nMAssay Description:Displacement of [3H]nicotinic acid from mouse GPR109a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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