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Found 30 Enz. Inhib. hit(s) with all data for entry = 3344
LigandPNGBDBM31647(tetrahydrobenzothiophene (THBT), 21)
Affinity DataIC50:  10nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31648(tetrahydrobenzothiophene (THBT), 22)
Affinity DataIC50:  25nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31637(tetrahydrobenzothiophene (THBT), 6)
Affinity DataIC50:  50nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
LigandPNGBDBM31644(tetrahydrobenzothiophene (THBT), 23)
Affinity DataIC50:  50nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31638(tetrahydrobenzothiophene (THBT), 13a)
Affinity DataIC50:  79nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31649(tetrahydrobenzothiophene (THBT), 24)
Affinity DataIC50:  100nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31648(tetrahydrobenzothiophene (THBT), 22)
Affinity DataIC50:  126nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31647(tetrahydrobenzothiophene (THBT), 21)
Affinity DataIC50:  126nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31636(tetrahydrobenzothiophene (THBT), 4)
Affinity DataIC50:  200nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31636(tetrahydrobenzothiophene (THBT), 4)
Affinity DataIC50:  316nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31650(tetrahydrobenzothiophene (THBT), 25)
Affinity DataIC50:  398nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31644(tetrahydrobenzothiophene (THBT), 23)
Affinity DataIC50:  398nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31637(tetrahydrobenzothiophene (THBT), 6)
Affinity DataIC50:  501nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31640(tetrahydrobenzothiophene (THBT), 14)
Affinity DataIC50:  631nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31646(tetrahydrobenzothiophene (THBT), 20)
Affinity DataIC50:  1.26E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31642(tetrahydrobenzothiophene (THBT), 16)
Affinity DataIC50:  1.26E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31650(tetrahydrobenzothiophene (THBT), 25)
Affinity DataIC50:  1.59E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31645(tetrahydrobenzothiophene (THBT), 19)
Affinity DataIC50:  2.00E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31649(tetrahydrobenzothiophene (THBT), 24)
Affinity DataIC50:  2.51E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31651(tetrahydrobenzothiophene (THBT), 18)
Affinity DataIC50:  2.51E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31641(tetrahydrobenzothiophene (THBT), 15)
Affinity DataIC50: >2.51E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31640(tetrahydrobenzothiophene (THBT), 14)
Affinity DataIC50: >2.51E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31641(tetrahydrobenzothiophene (THBT), 15)
Affinity DataIC50: >2.51E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31651(tetrahydrobenzothiophene (THBT), 18)
Affinity DataIC50:  5.01E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31643(tetrahydrobenzothiophene (THBT), 17)
Affinity DataIC50:  5.01E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31645(tetrahydrobenzothiophene (THBT), 19)
Affinity DataIC50:  6.31E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31642(tetrahydrobenzothiophene (THBT), 16)
Affinity DataIC50:  6.31E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31646(tetrahydrobenzothiophene (THBT), 20)
Affinity DataIC50:  6.31E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31639(tetrahydrobenzothiophene (THBT), 13b)
Affinity DataIC50: >1.00E+4nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM31643(tetrahydrobenzothiophene (THBT), 17)
Affinity DataIC50:  3.16E+4nMpH: 7.5 T: 2°CAssay Description:Inhibition of PDE4 is measured using a luminescence-coupled assay system developed by Cambrex. This assay system couples the formation of AMP, derive...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed