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Found 11 Enz. Inhib. hit(s) with all data for entry = 3356
TargetPteridine reductase(Trypanosoma brucei brucei)
University Of Dundee

LigandPNGBDBM31801(2-aminobenzimidazole deriv., 12)
Affinity DataKi:  7nM ΔG°:  -46.2kJ/molepH: 6.0 T: 2°CAssay Description:TbPTR1 activity was measured in 96-well microtiter plates via reduction of cytochrome c (cytc) as a result of the enzymatic production of tetrahydrob...More data for this Ligand-Target Pair
TargetPteridine reductase(Trypanosoma brucei brucei)
University Of Dundee

LigandPNGBDBM31800(2-aminobenzimidazole deriv., 11)
Affinity DataKi:  47nM ΔG°:  -41.5kJ/molepH: 6.0 T: 2°CAssay Description:TbPTR1 activity was measured in 96-well microtiter plates via reduction of cytochrome c (cytc) as a result of the enzymatic production of tetrahydrob...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPteridine reductase(Trypanosoma brucei brucei)
University Of Dundee

LigandPNGBDBM31798(2-aminobenzimidazole deriv., 9)
Affinity DataKi:  400nM ΔG°:  -36.3kJ/molepH: 6.0 T: 2°CAssay Description:TbPTR1 activity was measured in 96-well microtiter plates via reduction of cytochrome c (cytc) as a result of the enzymatic production of tetrahydrob...More data for this Ligand-Target Pair
TargetPteridine reductase(Trypanosoma brucei brucei)
University Of Dundee

LigandPNGBDBM31799(2-aminobenzimidazole deriv., 10)
Affinity DataKi:  510nM ΔG°:  -35.7kJ/molepH: 6.0 T: 2°CAssay Description:TbPTR1 activity was measured in 96-well microtiter plates via reduction of cytochrome c (cytc) as a result of the enzymatic production of tetrahydrob...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPteridine reductase(Trypanosoma brucei brucei)
University Of Dundee

LigandPNGBDBM31795(2-aminobenzimidazole deriv., 6)
Affinity DataKi:  9.80E+3nM ΔG°:  -28.4kJ/molepH: 6.0 T: 2°CAssay Description:TbPTR1 activity was measured in 96-well microtiter plates via reduction of cytochrome c (cytc) as a result of the enzymatic production of tetrahydrob...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPteridine reductase(Trypanosoma brucei brucei)
University Of Dundee

LigandPNGBDBM31794(2-aminobenzimidazole deriv., 4 | 5-Chloro-1H-benzo...)
Affinity DataKi:  1.06E+4nM ΔG°:  -28.2kJ/molepH: 6.0 T: 2°CAssay Description:TbPTR1 activity was measured in 96-well microtiter plates via reduction of cytochrome c (cytc) as a result of the enzymatic production of tetrahydrob...More data for this Ligand-Target Pair
TargetPteridine reductase(Trypanosoma brucei brucei)
University Of Dundee

LigandPNGBDBM31791(2-aminobenzothiazole deriv., 2)
Affinity DataKi:  2.11E+4nM ΔG°:  -26.5kJ/molepH: 6.0 T: 2°CAssay Description:TbPTR1 activity was measured in 96-well microtiter plates via reduction of cytochrome c (cytc) as a result of the enzymatic production of tetrahydrob...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPteridine reductase(Trypanosoma brucei brucei)
University Of Dundee

LigandPNGBDBM31797(2-aminobenzimidazole deriv., 8)
Affinity DataKi:  2.39E+4nM ΔG°:  -26.2kJ/molepH: 6.0 T: 2°CAssay Description:TbPTR1 activity was measured in 96-well microtiter plates via reduction of cytochrome c (cytc) as a result of the enzymatic production of tetrahydrob...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPteridine reductase(Trypanosoma brucei brucei)
University Of Dundee

LigandPNGBDBM31793(2-aminobenzothiazole deriv., 3)
Affinity DataKi:  1.41E+5nM ΔG°:  -21.8kJ/molepH: 6.0 T: 2°CAssay Description:TbPTR1 activity was measured in 96-well microtiter plates via reduction of cytochrome c (cytc) as a result of the enzymatic production of tetrahydrob...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPteridine reductase(Trypanosoma brucei brucei)
University Of Dundee

LigandPNGBDBM31796(2-aminobenzimidazole deriv., 7)
Affinity DataKi: >2.00E+5nM ΔG°: >-21.0kJ/molepH: 6.0 T: 2°CAssay Description:TbPTR1 activity was measured in 96-well microtiter plates via reduction of cytochrome c (cytc) as a result of the enzymatic production of tetrahydrob...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPteridine reductase(Trypanosoma brucei brucei)
University Of Dundee

LigandPNGBDBM7960(1H-1,3-benzodiazol-2-amine | 2-Aminobenzimidazole ...)
Affinity DataKi:  2.88E+5nM ΔG°:  -20.1kJ/molepH: 6.0 T: 2°CAssay Description:TbPTR1 activity was measured in 96-well microtiter plates via reduction of cytochrome c (cytc) as a result of the enzymatic production of tetrahydrob...More data for this Ligand-Target Pair