Compile Data Set for Download or QSAR
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Found 13 Enz. Inhib. hit(s) with all data for entry = 50030467
TargetAcid-sensing ion channel 3(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50296576(2-(3-chloro-5-methylphenyl)-1H-indole-5-carboximid...)
Affinity DataIC50:  5.10E+4nMAssay Description:Inhibition of ASIC3 by patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 3(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50296570(2-(3-bromo-5-fluorophenyl)-1H-indole-5-carboximida...)
Affinity DataIC50:  5.90E+4nMAssay Description:Inhibition of ASIC3 by patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 3(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50296571(2-(3,5-dibromophenyl)-1H-indole-5-carboximidamide ...)
Affinity DataIC50:  5.90E+4nMAssay Description:Inhibition of ASIC3 by patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 3(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50296575(2-(3-(benzylamino)-5-chlorophenyl)-1H-indole-5-car...)
Affinity DataIC50:  7.70E+4nMAssay Description:Inhibition of ASIC3 by patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 3(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50296573(2-(3-amino-5-chlorophenyl)-1H-indole-5-carboximida...)
Affinity DataIC50:  9.50E+4nMAssay Description:Inhibition of ASIC3 by patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 3(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50296574(2-(3-chloro-5-((phenylamino)methyl)phenyl)-1H-indo...)
Affinity DataIC50:  1.14E+5nMAssay Description:Inhibition of ASIC3 by patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 3(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50296565(2-(3,5-dichlorophenyl)-1H-indole-5-carboximidamide...)
Affinity DataIC50:  1.33E+5nMAssay Description:Inhibition of ASIC3 by patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 3(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50296566(2-(2,3,5-trichlorophenyl)-1H-indole-5-carboximidam...)
Affinity DataIC50:  1.35E+5nMAssay Description:Inhibition of ASIC3 by patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 3(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50296567(2-(3,5-dichloro-4-cyanophenyl)-1H-indole-5-carboxi...)
Affinity DataIC50:  2.72E+5nMAssay Description:Inhibition of ASIC3 by patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 3(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50296569(2-(3-chloro-5-fluorophenyl)-1H-indole-5-carboximid...)
Affinity DataIC50:  2.78E+5nMAssay Description:Inhibition of ASIC3 by patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 3(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50296568(2-(2,6-dichloropyridin-4-yl)-1H-indole-5-carboximi...)
Affinity DataIC50:  2.91E+5nMAssay Description:Inhibition of ASIC3 by patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 3(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50296572(2-(3-fluoro-5-methoxyphenyl)-1H-indole-5-carboximi...)
Affinity DataIC50:  3.74E+5nMAssay Description:Inhibition of ASIC3 by patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcid-sensing ion channel 3(Homo sapiens (Human))
Merck

Curated by ChEMBL
LigandPNGBDBM50287160(2-Phenyl-1H-indole-5-carboxamidine | 2-phenyl-1H-i...)
Affinity DataIC50:  2.77E+6nMAssay Description:Inhibition of ASIC3 by patch-clamp electrophysiology assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed