Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50004254
TargetIntegrase(Human immunodeficiency virus 1)
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50184349((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-1-(4-f...)
Affinity DataIC50:  17nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli BL21 (DE3) by gel based assay in presence of magnesiumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50480767(CHEMBL562899)
Affinity DataIC50:  30nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli BL21 (DE3) by gel based assay in presence of magnesiumMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50480768(CHEMBL559753)
Affinity DataIC50:  120nMAssay Description:Inhibition of HIV1 integrase strand transfer activity expressed in Escherichia coli BL21 (DE3) by gel based assay in presence of magnesiumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50184349((Z)-4-[6-((Z)-3-carboxy-3-hydroxy-acryloyl)-1-(4-f...)
Affinity DataIC50:  440nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli BL21 (DE3) by gel based assay in presence of magnesiumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50480767(CHEMBL562899)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli BL21 (DE3) by gel based assay in presence of magnesiumMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetIntegrase(Human immunodeficiency virus 1)
Facult£S Universitaires Notre-Dame De La Paix

Curated by ChEMBL
LigandPNGBDBM50480768(CHEMBL559753)
Affinity DataIC50:  7.80E+4nMAssay Description:Inhibition of HIV1 integrase 3'-processing activity expressed in Escherichia coli BL21 (DE3) by gel based assay in presence of magnesiumMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed