Compile Data Set for Download or QSAR
maximum 50k data
Found 34 Enz. Inhib. hit(s) with all data for entry = 50000825
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010259(Acetic acid 10,10b-dihydroxy-6-{2-[3-(4-hydroxy-ph...)
Affinity DataKd:  2.80E+3nMAssay Description:Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 1(Bos taurus)
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010261((3R,4aR,5S,6S,6aS,10S,10aR,10bS)-3-ethenyl-6,10,10...)
Affinity DataKd:  29nMAssay Description:Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010261((3R,4aR,5S,6S,6aS,10S,10aR,10bS)-3-ethenyl-6,10,10...)
Affinity DataKd:  5.00E+3nMAssay Description:Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010263(Acetic acid 10,10b-dihydroxy-6-(2-isothiocyanato-e...)
Affinity DataKd:  300nMAssay Description:Binding activity against Glucose transporter in human erythrocyte membrane using [125I]-7-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010262(CHEMBL326703 | {4-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 1(Bos taurus)
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010264((2-Isothiocyanato-ethyl)-carbamic acid 6,10,10b-tr...)
Affinity DataKd:  110nMAssay Description:Binding activity against Adenylate cyclase in bovine brain membrane using [125I]-6-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 1(Bos taurus)
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010259(Acetic acid 10,10b-dihydroxy-6-{2-[3-(4-hydroxy-ph...)
Affinity DataKd:  9nMAssay Description:Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 1(Bos taurus)
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010263(Acetic acid 10,10b-dihydroxy-6-(2-isothiocyanato-e...)
Affinity DataKd:  130nMAssay Description:Binding activity against Adenylate cyclase in bovine brain membrane using [125I]-6-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010265(CHEMBL327142 | {2-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  1.10E+3nMAssay Description:Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010266(CHEMBL324659 | {6-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  400nMAssay Description:Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 1(Bos taurus)
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010267(CHEMBL92719 | [2-(4-Hydroxy-phenyl)-ethyl]-carbami...)
Affinity DataKd:  236nMAssay Description:Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010267(CHEMBL92719 | [2-(4-Hydroxy-phenyl)-ethyl]-carbami...)
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010268((2-Amino-ethyl)-carbamic acid (3R,4aR,5S,6S,6aS,10...)
Affinity DataKd:  2.80E+4nMAssay Description:Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 1(Bos taurus)
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010269(CHEMBL327672 | [2-(4-Hydroxy-phenyl)-ethyl]-carbam...)
Affinity DataKd:  61nMAssay Description:Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010264((2-Isothiocyanato-ethyl)-carbamic acid 6,10,10b-tr...)
Affinity DataKd:  500nMAssay Description:Binding activity against Glucose transporter in human erythrocyte membrane using [125I]-7-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 1(Bos taurus)
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010270(Acetic acid 6-[2-(2-bromo-acetylamino)-ethylcarbam...)
Affinity DataKd:  10nMAssay Description:Binding activity against Adenylate cyclase in bovine brain membrane using [125I]-6-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 1(Bos taurus)
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010272(CHEMBL322952 | {6-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  94nMAssay Description:Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 1(Bos taurus)
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010271(CHEMBL111425 | {4-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  60nMAssay Description:Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010273(CHEMBL111738 | {7-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  100nMAssay Description:Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010271(CHEMBL111425 | {4-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  800nMAssay Description:Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010274(Acetic acid (3R,4aR,5S,6S,6aS,10S,10aR,10bS)-6-(2-...)
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 1(Bos taurus)
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010266(CHEMBL324659 | {6-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  82nMAssay Description:Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 1(Bos taurus)
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010273(CHEMBL111738 | {7-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  53nMAssay Description:Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010270(Acetic acid 6-[2-(2-bromo-acetylamino)-ethylcarbam...)
Affinity DataKd:  1.70E+4nMAssay Description:Binding activity against Glucose transporter in human erythrocyte membrane using [125I]-7-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 1(Bos taurus)
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010274(Acetic acid (3R,4aR,5S,6S,6aS,10S,10aR,10bS)-6-(2-...)
Affinity DataKd:  34nMAssay Description:Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010260(CHEMBL107566 | [2-(2-Bromo-acetylamino)-ethyl]-car...)
Affinity DataKd:  1.30E+3nMAssay Description:Binding activity against Glucose transporter in human erythrocyte membrane using [125I]-7-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010272(CHEMBL322952 | {6-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 1(Bos taurus)
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010265(CHEMBL327142 | {2-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  13nMAssay Description:Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010275(CHEMBL324463 | {2-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd: >1.00E+5nMAssay Description:Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSolute carrier family 2, facilitated glucose transporter member 1(Homo sapiens (Human))
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010269(CHEMBL327672 | [2-(4-Hydroxy-phenyl)-ethyl]-carbam...)
Affinity DataKd:  240nMAssay Description:Inhibition of [125I]-7-IHPP-Fsk binding to glucose transporter of human erythrocyte membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 1(Bos taurus)
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010275(CHEMBL324463 | {2-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  174nMAssay Description:Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 1(Bos taurus)
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010262(CHEMBL326703 | {4-[3-(4-Hydroxy-phenyl)-propionyla...)
Affinity DataKd:  80nMAssay Description:Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 1(Bos taurus)
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010268((2-Amino-ethyl)-carbamic acid (3R,4aR,5S,6S,6aS,10...)
Affinity DataKd:  98nMAssay Description:Displacement of [125I]-6-IHPP-Fsk from adenylate cyclase of bovine brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenylate cyclase type 1(Bos taurus)
Food And Drug Administration

Curated by ChEMBL
LigandPNGBDBM50010260(CHEMBL107566 | [2-(2-Bromo-acetylamino)-ethyl]-car...)
Affinity DataKd:  10nMAssay Description:Binding activity against Adenylate cyclase in bovine brain membrane using [125I]-6-IHPP-Fsk as the radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed