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Found 102 Enz. Inhib. hit(s) with all data for entry = 50030705
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50132713(Arachidonic acid derivative | CHEMBL113262 | Methy...)
Affinity DataIC50:  0.330nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM60622(BDBM50300355 | US11753371, Compound JZL-184 | US91...)
Affinity DataIC50:  6nMAssay Description:Inhibition of human MGLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50059523((6Z,9Z,12Z,15Z)-1,1,1-trifluorohenicosa-6,9,12,15-...)
Affinity DataIC50:  12.3nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50132713(Arachidonic acid derivative | CHEMBL113262 | Methy...)
Affinity DataIC50:  26.3nMAssay Description:Inhibition of human MGLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM26736(CHEMBL509860 | LY2183240 | N,N-dimethyl-5-[(4-phen...)
Affinity DataIC50:  37.3nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM26736(CHEMBL509860 | LY2183240 | N,N-dimethyl-5-[(4-phen...)
Affinity DataIC50:  54.4nMAssay Description:Inhibition of human MGLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300344(1-Biphenyl-4-ylmethylmaleimide | CHEMBL576859)
Affinity DataIC50:  790nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300346(CHEMBL566336 | N-Oleylmaleimide)
Affinity DataIC50:  930nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM60419(BDBM50295658 | NAM)
Affinity DataIC50:  1.12E+3nMAssay Description:Inhibition of human MGLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300339(1-Biphenyl-2-ylmaleimide | CHEMBL567440)
Affinity DataIC50:  1.55E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300341(1-Biphenyl-4-ylmaleimide | CHEMBL567545)
Affinity DataIC50:  1.62E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300351((1-(6-(2,5-dioxo-2H-pyrrol-1(5H)-yl)-hexyl)-1H-mal...)
Affinity DataIC50:  1.70E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300349(1,4-bis(malimido)xylene | CHEMBL565711)
Affinity DataIC50:  1.70E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300352(1,8-bis-maleimidodiethyleneglycol | CHEMBL575383)
Affinity DataIC50:  1.95E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300316(1-(2-Ethylphenyl)maleimide | CHEMBL574140)
Affinity DataIC50:  2.00E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300347(CHEMBL573689 | phenyl-1,3-bismaleimide)
Affinity DataIC50:  2.03E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300322(1-(4-Heptylphenyl)maleimide | CHEMBL565892)
Affinity DataIC50:  2.12E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300342(1-(4-Phenylbutyl)maleimide | 1-(4-phenylbutyl)-1H-...)
Affinity DataIC50:  2.14E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM60419(BDBM50295658 | NAM)
Affinity DataIC50:  2.18E+3nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300348(CHEMBL576594 | phenyl-1,4-bismaleimide)
Affinity DataIC50:  2.22E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50270000(1,1-(Methylene-di-1,4-phenylene)-bismaleimide | 1,...)
Affinity DataIC50:  2.24E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300337(1-(3-Iodophenyl)maleimide | CHEMBL565710)
Affinity DataIC50:  2.24E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300340(1-Biphenyl-3-ylmaleimide | CHEMBL567622 | cid_9309...)
Affinity DataIC50:  2.34E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300328(1-(3-Fluorophenyl)maleimide | CHEMBL574358)
Affinity DataIC50:  2.39E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300313(1-(2-Methylphenyl)maleimide | CHEMBL578794)
Affinity DataIC50:  2.69E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300345(CHEMBL568289 | N-Palmitylmaleimide)
Affinity DataIC50:  2.69E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300314(1-(3-Methylphenyl)maleimide | CHEMBL567421)
Affinity DataIC50:  2.75E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300318(1-(4-Ethylphenyl)maleimide | CHEMBL577071)
Affinity DataIC50:  2.82E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300331(1-(3-Chlorophenyl)maleimide | CHEMBL578977)
Affinity DataIC50:  2.82E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300321(1-(4-Isopropylphenyl)maleimide | CHEMBL576625)
Affinity DataIC50:  2.88E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300333(1-(2-Bromophenyl)maleimide | CHEMBL578978)
Affinity DataIC50:  2.92E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300343(1-(4-Ethylbenzyl)maleimide | CHEMBL576626)
Affinity DataIC50:  3.55E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50050711(1-Nonyl-pyrrole-2,5-dione | CHEMBL47299 | N-Nonylm...)
Affinity DataIC50:  3.55E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM60622(BDBM50300355 | US11753371, Compound JZL-184 | US91...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300330(1-(2-Chlorophenyl)maleimide | CHEMBL565700)
Affinity DataIC50:  4.17E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300334(1-(3-Bromophenyl)maleimide | CHEMBL583957)
Affinity DataIC50:  4.27E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300338(1-(4-Iodophenyl)maleimide | CHEMBL579183)
Affinity DataIC50:  4.34E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300335(1-(4-Bromophenyl)maleimide | CHEMBL566998)
Affinity DataIC50:  4.37E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300327(1-(2-Fluorophenyl)maleimide | CHEMBL579012)
Affinity DataIC50:  4.47E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300317(1-(3-Ethylphenyl)maleimide | CHEMBL568527)
Affinity DataIC50:  4.68E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300336(1-(2-Iodophenyl)maleimide | CHEMBL566999)
Affinity DataIC50:  5.01E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM7804(1-benzyl-2,5-dihydro-1H-pyrrole-2,5-dione | Maleim...)
Affinity DataIC50:  5.14E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300329(1-(4-Fluorophenyl)maleimide | CHEMBL583956)
Affinity DataIC50:  5.18E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50128581(Biphenyl-3-yl-carbamic acid cyclohexyl ester | CHE...)
Affinity DataIC50:  5.65E+3nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300326(1-(4-Methoxyphenyl)maleimide | CHEMBL568288)
Affinity DataIC50:  5.75E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300341(1-Biphenyl-4-ylmaleimide | CHEMBL567545)
Affinity DataIC50:  5.89E+3nMAssay Description:Displacement of [3H]ethanolamine from human recombinant FAAH by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300319(1-(4-Propylphenyl)maleimide | CHEMBL568528)
Affinity DataIC50:  5.89E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50059523((6Z,9Z,12Z,15Z)-1,1,1-trifluorohenicosa-6,9,12,15-...)
Affinity DataIC50:  6.31E+3nMAssay Description:Inhibition of human MGLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300325(1-(3-Methoxyphenyl)maleimide | CHEMBL566111)
Affinity DataIC50:  6.60E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Louvain Drug Research Institute

Curated by ChEMBL
LigandPNGBDBM50300324(1-(2-Methoxyphenyl)maleimide | CHEMBL565904)
Affinity DataIC50:  6.92E+3nMAssay Description:Displacement of [3H]2-OG from human MGL by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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