Compile Data Set for Download or QSAR
maximum 50k data
Found 26 Enz. Inhib. hit(s) with all data for entry = 50038874
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM18207((1R,2S,10S,11S,13R,14R,15S,17S)-1-fluoro-14,17-dih...)
Affinity DataIC50:  5nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294138(CHEMBL524378 | N-(5-(2-(3-(2-(2-((8R,9S,10R,11R,13...)
Affinity DataIC50:  5.70nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294160(CHEMBL552770 | N-(1-((8S,9R,10S,11S,13S,14S,16R,17...)
Affinity DataIC50:  8.30nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294146(CHEMBL539699 | N-(5-(1-((8S,9R,10S,11S,13S,14S,16R...)
Affinity DataIC50:  8.5nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294153(3-acetamido-N-(1-((8S,9R,10S,11S,13S,14S,16R,17R)-...)
Affinity DataIC50:  9.30nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294159(CHEMBL553019 | N-(2-(3-(2-(2-((8S,9R,10S,11S,13S,1...)
Affinity DataIC50:  9.80nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294147(CHEMBL537949 | N-(5-(5-(1-((8S,9R,10S,11S,13S,14S,...)
Affinity DataIC50:  12nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294139(CHEMBL540936 | N-(5-(5-(2-(3-(2-(2-((8R,9S,10R,11R...)
Affinity DataIC50:  14nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294137(CHEMBL556523)
Affinity DataIC50:  14nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294157(1-(2-(2-((8S,9R,10S,11S,13S,14S,16R,17R)-9-fluoro-...)
Affinity DataIC50:  15nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294149(CHEMBL553440 | N-(5-(5-(5-(5-(1-((8S,9R,10S,11S,13...)
Affinity DataIC50:  16nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294150(CHEMBL556793 | N-(4-(5-(5-(5-(5-(1-((8S,9R,10S,11S...)
Affinity DataIC50:  16nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294148(CHEMBL563289 | N-(5-(5-(5-(1-((8S,9R,10S,11S,13S,1...)
Affinity DataIC50:  20nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294152(CHEMBL563739)
Affinity DataIC50:  20nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294144(CHEMBL553018 | N-(5-(5-(4-(5-(5-(5-(5-(2-(3-(2-(2-...)
Affinity DataIC50:  21nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294143(CHEMBL551944 | N-(5-(4-(5-(5-(5-(5-(2-(3-(2-(2-((8...)
Affinity DataIC50:  21nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294151(CHEMBL552769 | N-(5-(4-(5-(5-(5-(5-(1-((8S,9R,10S,...)
Affinity DataIC50:  22nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294142(CHEMBL540184 | N-(4-(5-(5-(5-(5-(2-(3-(2-(2-((8R,9...)
Affinity DataIC50:  23nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294140(CHEMBL538939 | N-(5-(5-(5-(2-(3-(2-(2-((8R,9S,10R,...)
Affinity DataIC50:  26nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294145(CHEMBL564923)
Affinity DataIC50:  27nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294141(CHEMBL541765 | N-(5-(5-(5-(5-(2-(3-(2-(2-((8R,9S,1...)
Affinity DataIC50:  34nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294158(CHEMBL554774 | N-(5-(2-((8R,9S,10R,11R,13R,14R,16S...)
Affinity DataIC50:  460nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294154(CHEMBL557958 | N-(5-(5-(2-((8R,9S,10R,11R,13R,14R,...)
Affinity DataIC50:  480nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294155(CHEMBL553441 | N-(5-(5-(5-(2-((8R,9S,10R,11R,13R,1...)
Affinity DataIC50:  550nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50271344((8S,9R,10S,11S,13S,14S,16R,17R)-9-fluoro-11,17-dih...)
Affinity DataIC50:  600nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of Texas Southwestern Medical Center

Curated by ChEMBL
LigandPNGBDBM50294156(CHEMBL556536 | N-(5-(5-(5-(4-(5-(5-(5-(5-(2-((8R,9...)
Affinity DataIC50:  840nMAssay Description:Displacement of fluormone from human recombinant glucocorticoid receptor ligand binding domain by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed