Compile Data Set for Download or QSAR
maximum 50k data
Found 31 Enz. Inhib. hit(s) with all data for entry = 50004276
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481036(CHEMBL568589)
Affinity DataIC50:  0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481029(CHEMBL569671)
Affinity DataIC50:  0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481028(CHEMBL566620)
Affinity DataIC50:  0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481018(CHEMBL568883)
Affinity DataIC50:  0.302nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481014(CHEMBL568951)
Affinity DataIC50:  0.339nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481023(CHEMBL566849)
Affinity DataIC50:  0.398nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481020(CHEMBL565964)
Affinity DataIC50:  0.398nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481040(CHEMBL566842)
Affinity DataIC50:  0.501nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481024(CHEMBL566902)
Affinity DataIC50:  0.741nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481017(CHEMBL568840)
Affinity DataIC50:  0.794nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481015(CHEMBL568832)
Affinity DataIC50:  0.794nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481025(CHEMBL567444)
Affinity DataIC50:  0.851nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481033(CHEMBL565528)
Affinity DataIC50:  0.891nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481035(CHEMBL569670)
Affinity DataIC50:  1nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481037(CHEMBL569236)
Affinity DataIC50:  1.30nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481032(CHEMBL569569)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481022(CHEMBL568365)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM586099(BDBM50064200 | TL-3)
Affinity DataIC50:  2nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481019(CHEMBL571731)
Affinity DataIC50:  2.20nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481031(CHEMBL567043)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481041(CHEMBL569673)
Affinity DataIC50:  3.20nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481016(CHEMBL568817)
Affinity DataIC50:  4nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481038(CHEMBL568977)
Affinity DataIC50:  4nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM198((2S)-N-[(2S,3S,4S,5S)-3,4-dihydroxy-5-[(2S)-3-meth...)
Affinity DataIC50:  15nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481027(CHEMBL566839)
Affinity DataIC50:  18nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481030(CHEMBL570827)
Affinity DataIC50:  22nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481013(CHEMBL569111)
Affinity DataIC50:  38nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481034(CHEMBL567500)
Affinity DataIC50:  100nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481021(CHEMBL565766)
Affinity DataIC50:  141nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481039(CHEMBL569672)
Affinity DataIC50:  339nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Universidade Federal De Lavras

Curated by ChEMBL
LigandPNGBDBM50481026(CHEMBL569573)
Affinity DataIC50:  363nMAssay Description:Inhibition of HIV1 protease expressed in Escherichia coli K12 assessed as inhibition of enzyme activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed