Compile Data Set for Download or QSAR
maximum 50k data
Found 44 Enz. Inhib. hit(s) with all data for entry = 50030503
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297219(1-(4-tert-butylphenylsulfonyl)-4-methoxy-4-methyla...)
Affinity DataIC50:  3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297216(1-(4-tert-butylphenylsulfonyl)-4-methylazepan-4-ol...)
Affinity DataIC50:  5nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297220(1-(4-tert-butylphenylsulfonyl)-4-methoxyazepane | ...)
Affinity DataIC50:  7nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297203((4-methoxyphenyl)(4-phenylazepan-1-yl)methanone | ...)
Affinity DataIC50:  9nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297217(1-(4-tert-butylphenylsulfonyl)-4-cyclopropylazepan...)
Affinity DataIC50:  12nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297223(4-methoxy-1-(4-(2-methoxypropan-2-yl)phenylsulfony...)
Affinity DataIC50:  20nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297216(1-(4-tert-butylphenylsulfonyl)-4-methylazepan-4-ol...)
Affinity DataIC50:  35nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297221(1-(4-tert-butylphenylsulfonyl)-4-cyclopropyl-4-met...)
Affinity DataIC50:  43nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297219(1-(4-tert-butylphenylsulfonyl)-4-methoxy-4-methyla...)
Affinity DataIC50:  57nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297204((E)-1-(4-methoxyphenylsulfonyl)-4-phenyl-2,3,6,7-t...)
Affinity DataIC50:  58nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297205((E)-1-(4-tert-butylphenylsulfonyl)-4-phenyl-2,3,6,...)
Affinity DataIC50:  68nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297206((E)-4-phenyl-1-tosyl-2,3,6,7-tetrahydro-1H-azepine...)
Affinity DataIC50:  76nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297207((E)-1-(4-ethylphenylsulfonyl)-4-phenyl-2,3,6,7-tet...)
Affinity DataIC50:  97nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297222(1-(4-tert-butylphenylsulfonyl)-4-methoxy-4-phenyla...)
Affinity DataIC50:  110nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297203((4-methoxyphenyl)(4-phenylazepan-1-yl)methanone | ...)
Affinity DataIC50:  111nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297224(2-(4-(4-methoxy-4-methylazepan-1-ylsulfonyl)phenyl...)
Affinity DataIC50:  113nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297217(1-(4-tert-butylphenylsulfonyl)-4-cyclopropylazepan...)
Affinity DataIC50:  115nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297209((E)-5-phenyl-1-tosyl-2,3,4,7-tetrahydro-1H-azepine...)
Affinity DataIC50:  124nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297220(1-(4-tert-butylphenylsulfonyl)-4-methoxyazepane | ...)
Affinity DataIC50:  165nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297210((E)-1-(4-methoxyphenylsulfonyl)-5-phenyl-2,3,4,7-t...)
Affinity DataIC50:  178nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297222(1-(4-tert-butylphenylsulfonyl)-4-methoxy-4-phenyla...)
Affinity DataIC50:  210nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297223(4-methoxy-1-(4-(2-methoxypropan-2-yl)phenylsulfony...)
Affinity DataIC50:  229nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297212(1-(4-tert-butylphenylsulfonyl)-4-phenylazepan-4-ol...)
Affinity DataIC50:  307nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297221(1-(4-tert-butylphenylsulfonyl)-4-cyclopropyl-4-met...)
Affinity DataIC50:  328nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297211((E)-1-(4-tert-butylphenylsulfonyl)-5-phenyl-2,3,4,...)
Affinity DataIC50:  358nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297218(1-(4-tert-butylphenylsulfonyl)azepan-4-ol | CHEMBL...)
Affinity DataIC50:  466nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297213(1-(4-ethylphenylsulfonyl)-4-phenylazepan-4-ol | CH...)
Affinity DataIC50:  493nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297218(1-(4-tert-butylphenylsulfonyl)azepan-4-ol | CHEMBL...)
Affinity DataIC50:  629nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297224(2-(4-(4-methoxy-4-methylazepan-1-ylsulfonyl)phenyl...)
Affinity DataIC50:  656nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297212(1-(4-tert-butylphenylsulfonyl)-4-phenylazepan-4-ol...)
Affinity DataIC50:  860nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297205((E)-1-(4-tert-butylphenylsulfonyl)-4-phenyl-2,3,6,...)
Affinity DataIC50:  905nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297208((E)-1-(2,4-dichlorophenylsulfonyl)-4-phenyl-2,3,6,...)
Affinity DataIC50:  994nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297214(1-(4-chlorophenylsulfonyl)-4-phenylazepan-4-ol | C...)
Affinity DataIC50:  1.07E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297207((E)-1-(4-ethylphenylsulfonyl)-4-phenyl-2,3,6,7-tet...)
Affinity DataIC50:  1.24E+3nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297208((E)-1-(2,4-dichlorophenylsulfonyl)-4-phenyl-2,3,6,...)
Affinity DataIC50:  1.28E+3nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297215(1-(4-methoxyphenylsulfonyl)-4-phenylazepan-4-ol | ...)
Affinity DataIC50:  1.32E+3nMAssay Description:Inhibition of human 11beta-HSD1 expressed in Sf9 cells by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297213(1-(4-ethylphenylsulfonyl)-4-phenylazepan-4-ol | CH...)
Affinity DataIC50:  1.41E+3nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297209((E)-5-phenyl-1-tosyl-2,3,4,7-tetrahydro-1H-azepine...)
Affinity DataIC50:  1.51E+3nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297206((E)-4-phenyl-1-tosyl-2,3,6,7-tetrahydro-1H-azepine...)
Affinity DataIC50:  1.55E+3nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297210((E)-1-(4-methoxyphenylsulfonyl)-5-phenyl-2,3,4,7-t...)
Affinity DataIC50:  1.55E+3nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297211((E)-1-(4-tert-butylphenylsulfonyl)-5-phenyl-2,3,4,...)
Affinity DataIC50:  1.65E+3nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297204((E)-1-(4-methoxyphenylsulfonyl)-4-phenyl-2,3,6,7-t...)
Affinity DataIC50:  1.88E+3nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297215(1-(4-methoxyphenylsulfonyl)-4-phenylazepan-4-ol | ...)
Affinity DataIC50:  1.98E+3nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target11-beta-hydroxysteroid dehydrogenase 1(Mus musculus (mouse))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50297214(1-(4-chlorophenylsulfonyl)-4-phenylazepan-4-ol | C...)
Affinity DataIC50:  2.72E+3nMAssay Description:Inhibition of mouse 11beta-HSD1 by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed