Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM22885![]() (3-[(2S)-1-(1H-imidazol-5-yl)propan-2-yl]-2-(2-{[(5...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 40 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonistic activity at histamine H3 receptor in rat cerebral cortex and is represented as Ki | J Med Chem 33: 4-11 (1990) Article DOI: 10.1021/jm00163a001 BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM85411![]() (GT 2174) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | PC cid PC sid UniChem Patents Similars | Article PubMed | 50 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonist activity against histamine H3 receptor and is represented as -log Ki. | J Med Chem 33: 4-11 (1990) Article DOI: 10.1021/jm00163a001 BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM22886![]() (3-[(2R)-1-(1H-imidazol-5-yl)propan-2-yl]-2-(2-{[(5...) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 60 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonistic activity at histamine H3 receptor in rat cerebral cortex and is represented as Ki. | J Med Chem 33: 4-11 (1990) Article DOI: 10.1021/jm00163a001 BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50406098![]() (CHEMBL12494) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 79 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonist activity against Histamine H3 receptor and represented as KB. | J Med Chem 33: 4-11 (1990) Article DOI: 10.1021/jm00163a001 BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50406100![]() (CHEMBL12459) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 200 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonist activity against Histamine H3 receptor and represented as KB. | J Med Chem 33: 4-11 (1990) Article DOI: 10.1021/jm00163a001 BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50406095![]() (CHEMBL275090) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem | Article PubMed | 631 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonist activity against histamine H3 receptor and is represented as -log Ki. | J Med Chem 33: 4-11 (1990) Article DOI: 10.1021/jm00163a001 BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50406101![]() (CHEMBL12550) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 631 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonist activity against Histamine H3 receptor and represented as KB. | J Med Chem 33: 4-11 (1990) Article DOI: 10.1021/jm00163a001 BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50406099![]() (CHEMBL416338) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem | Article PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonist activity against histamine H3 receptor and is represented as -log Ki. | J Med Chem 33: 4-11 (1990) Article DOI: 10.1021/jm00163a001 BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50406097![]() (CHEMBL12551) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonist activity against histamine H3 receptor and is represented as -log Ki. | J Med Chem 33: 4-11 (1990) Article DOI: 10.1021/jm00163a001 BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50406093![]() (CHEMBL276903) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | CHEMBL PC cid PC sid UniChem | Article PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonist activity against Histamine H3 receptor and represented as KB. | J Med Chem 33: 4-11 (1990) Article DOI: 10.1021/jm00163a001 BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Histamine H3 receptor (Rattus norvegicus (rat)) | BDBM50406096![]() (CHEMBL12025) | Reactome pathway KEGG UniProtKB/SwissProt GoogleScholar | Purchase CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.00E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Vrije Universiteit Curated by ChEMBL | Assay Description Evaluated for antagonist activity against Histamine H3 receptor and represented as KB. | J Med Chem 33: 4-11 (1990) Article DOI: 10.1021/jm00163a001 BindingDB Entry DOI: 10.7270/Q2GB230D | |||||||||||
More data for this Ligand-Target Pair |