Compile Data Set for Download or QSAR
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Found 30 Enz. Inhib. hit(s) with all data for entry = 50041785
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415502(CHEMBL598126)
Affinity DataEC50:  27nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415531(CHEMBL592297)
Affinity DataEC50:  23nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415504(CHEMBL596909)
Affinity DataEC50:  91nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415505(CHEMBL603662)
Affinity DataEC50:  160nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415506(CHEMBL599781)
Affinity DataEC50:  53nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415507(CHEMBL604937)
Affinity DataEC50:  28nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415508(CHEMBL599365)
Affinity DataEC50:  160nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415509(CHEMBL599164)
Affinity DataEC50:  25nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415510(CHEMBL591203)
Affinity DataEC50:  98nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415511(CHEMBL598553)
Affinity DataEC50:  21nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415512(CHEMBL603667)
Affinity DataEC50:  2.08E+3nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415513(CHEMBL597329)
Affinity DataEC50:  570nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415514(CHEMBL597330)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415515(CHEMBL603874)
Affinity DataEC50:  2.70E+3nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415516(CHEMBL599374)
Affinity DataEC50:  28nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415517(CHEMBL599375)
Affinity DataEC50:  62nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415518(CHEMBL608156)
Affinity DataEC50:  710nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415519(CHEMBL591677)
Affinity DataEC50: >1.00E+4nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415520(CHEMBL599376)
Affinity DataEC50:  49nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415521(CHEMBL609624)
Affinity DataEC50:  44nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415522(CHEMBL597341)
Affinity DataEC50:  220nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415523(CHEMBL597342)
Affinity DataEC50:  5.57E+3nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415524(CHEMBL597544)
Affinity DataEC50:  6.73E+3nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415525(CHEMBL589667)
Affinity DataEC50:  100nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415526(CHEMBL591302)
Affinity DataEC50:  44nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415527(CHEMBL592146)
Affinity DataEC50:  260nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415528(CHEMBL602304)
Affinity DataEC50:  500nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415529(CHEMBL589898)
Affinity DataEC50:  29nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415530(CHEMBL602305)
Affinity DataEC50:  95nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily KQT member 2/3(Homo sapiens (Human))
Icagen

Curated by ChEMBL
LigandPNGBDBM50415503(CHEMBL603661)
Affinity DataEC50:  380nMAssay Description:Activation of KCNQ2/KCNQ3 expressed in CHO cells by isotopic efflux assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed