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Found 29 Enz. Inhib. hit(s) with all data for entry = 50031214
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309063(2-(4-(methylsulfonyl)phenyl)-11-phenyl-4,9-dioxa-3...)
Affinity DataEC50:  1.90E+3nMAssay Description:Agonist activity at human full length PPARgamma expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309077(11-phenyl-2-(4-(trifluoromethyl)phenyl)-4,9-dioxa-...)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at human full length PPARgamma expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309065(2-(biphenyl-3-yl)-11-phenyl-4,9-dioxa-3,10-diazate...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human full length PPARgamma expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309066(2-(naphthalen-2-yl)-11-phenyl-4,9-dioxa-3,10-diaza...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human full length PPARgamma expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309067(11-phenyl-2-(5,6,7,8-tetrahydronaphthalen-2-yl)-4,...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human full length PPARgamma expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309068(2-(3,4-dimethoxyphenyl)-11-phenyl-4,9-dioxa-3,10-d...)
Affinity DataEC50:  800nMAssay Description:Agonist activity at human full length PPARgamma expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309069(2-(3,4-dimethylphenyl)-11-phenyl-4,9-dioxa-3,10-di...)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human full length PPARgamma expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309070(2-(3-methoxy-4-methylphenyl)-11-phenyl-4,9-dioxa-3...)
Affinity DataEC50:  1.60E+3nMAssay Description:Agonist activity at human full length PPARgamma expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309071(2-(4-fluoro-3-methoxyphenyl)-11-phenyl-4,9-dioxa-3...)
Affinity DataEC50:  700nMAssay Description:Agonist activity at human full length PPARgamma expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309072(CHEMBL592054 | IMIGLITAZAR)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human full length PPARgamma expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309073(2,11-diphenyl-4,9-dioxa-3,10-diazatetradeca-2,10-d...)
Affinity DataEC50:  2.30E+3nMAssay Description:Agonist activity at human full length PPARalpha expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309074(2-(4-fluorophenyl)-11-phenyl-4,9-dioxa-3,10-diazat...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human full length PPARalpha expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309075(11-phenyl-2-p-tolyl-4,9-dioxa-3,10-diazatetradeca-...)
Affinity DataEC50:  50nMAssay Description:Agonist activity at human full length PPARalpha expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309076(2-(4-methoxyphenyl)-11-phenyl-4,9-dioxa-3,10-diaza...)
Affinity DataEC50:  10nMAssay Description:Agonist activity at human full length PPARalpha expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309077(11-phenyl-2-(4-(trifluoromethyl)phenyl)-4,9-dioxa-...)
Affinity DataEC50:  400nMAssay Description:Agonist activity at human full length PPARalpha expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309063(2-(4-(methylsulfonyl)phenyl)-11-phenyl-4,9-dioxa-3...)
Affinity DataEC50:  2.40E+3nMAssay Description:Agonist activity at human full length PPARalpha expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309064(2-(3-butylphenyl)-11-phenyl-4,9-dioxa-3,10-diazate...)
Affinity DataEC50:  500nMAssay Description:Agonist activity at human full length PPARalpha expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309065(2-(biphenyl-3-yl)-11-phenyl-4,9-dioxa-3,10-diazate...)
Affinity DataEC50:  20nMAssay Description:Agonist activity at human full length PPARalpha expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309066(2-(naphthalen-2-yl)-11-phenyl-4,9-dioxa-3,10-diaza...)
Affinity DataEC50:  30nMAssay Description:Agonist activity at human full length PPARalpha expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309067(11-phenyl-2-(5,6,7,8-tetrahydronaphthalen-2-yl)-4,...)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human full length PPARalpha expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309068(2-(3,4-dimethoxyphenyl)-11-phenyl-4,9-dioxa-3,10-d...)
Affinity DataEC50:  100nMAssay Description:Agonist activity at human full length PPARalpha expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309069(2-(3,4-dimethylphenyl)-11-phenyl-4,9-dioxa-3,10-di...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human full length PPARalpha expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309070(2-(3-methoxy-4-methylphenyl)-11-phenyl-4,9-dioxa-3...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human full length PPARalpha expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309071(2-(4-fluoro-3-methoxyphenyl)-11-phenyl-4,9-dioxa-3...)
Affinity DataEC50:  400nMAssay Description:Agonist activity at human full length PPARalpha expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309072(CHEMBL592054 | IMIGLITAZAR)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human full length PPARalpha expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309074(2-(4-fluorophenyl)-11-phenyl-4,9-dioxa-3,10-diazat...)
Affinity DataEC50:  1.40E+3nMAssay Description:Agonist activity at human full length PPARgamma expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309075(11-phenyl-2-p-tolyl-4,9-dioxa-3,10-diazatetradeca-...)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at human full length PPARgamma expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309076(2-(4-methoxyphenyl)-11-phenyl-4,9-dioxa-3,10-diaza...)
Affinity DataEC50:  1.10E+3nMAssay Description:Agonist activity at human full length PPARgamma expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Zydus Research Centre

Curated by ChEMBL
LigandPNGBDBM50309064(2-(3-butylphenyl)-11-phenyl-4,9-dioxa-3,10-diazate...)
Affinity DataEC50:  200nMAssay Description:Agonist activity at human full length PPARgamma expressed in human HepG2 cells cotransfected with PPRE3-TK-luc assessed as induction of beta-galactos...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed