Compile Data Set for Download or QSAR
maximum 50k data
Found 17 Enz. Inhib. hit(s) with all data for entry = 50031753
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50318416(7alpha-(1-Hydroxy-1-methyl-ethyl)-6-phenyl-6-demet...)
Affinity DataIC50:  0.110nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor from Wistar rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50318412(7alpha-(1-Hydroxy-1-methyl-ethyl)-6-propoxy-6-deme...)
Affinity DataIC50:  0.130nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor from Wistar rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50318415(7alpha-(1-Hydroxy-1-methyl-ethyl)-6-(cyclopropylme...)
Affinity DataIC50:  0.140nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor from Wistar rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50318413(7alpha-(1-Hydroxy-1-methyl-ethyl)-6-ethoxy-6-demet...)
Affinity DataIC50:  0.180nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor from Wistar rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50318414(7alpha-(1-Hydroxy-1-methyl-ethyl)-6,7,8,14-tetrahy...)
Affinity DataIC50:  0.540nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor from Wistar rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  5.64nMAssay Description:Displacement of [3H]DAMGO from mu opioid receptor from Wistar rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50318413(7alpha-(1-Hydroxy-1-methyl-ethyl)-6-ethoxy-6-demet...)
Affinity DataIC50:  230nMAssay Description:Displacement of [3H]deltorphin-2 from delta opioid receptor from Wistar rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50318412(7alpha-(1-Hydroxy-1-methyl-ethyl)-6-propoxy-6-deme...)
Affinity DataIC50:  320nMAssay Description:Displacement of [3H]deltorphin-2 from delta opioid receptor from Wistar rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataIC50:  404nMAssay Description:Displacement of [3H]deltorphin-2 from delta opioid receptor from Wistar rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50318416(7alpha-(1-Hydroxy-1-methyl-ethyl)-6-phenyl-6-demet...)
Affinity DataIC50:  440nMAssay Description:Displacement of [3H]deltorphin-2 from delta opioid receptor from Wistar rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50318415(7alpha-(1-Hydroxy-1-methyl-ethyl)-6-(cyclopropylme...)
Affinity DataIC50:  650nMAssay Description:Displacement of [3H]deltorphin-2 from delta opioid receptor from Wistar rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50318414(7alpha-(1-Hydroxy-1-methyl-ethyl)-6,7,8,14-tetrahy...)
Affinity DataIC50:  1.35E+3nMAssay Description:Displacement of [3H]deltorphin-2 from delta opioid receptor from Wistar rat brain by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50318414(7alpha-(1-Hydroxy-1-methyl-ethyl)-6,7,8,14-tetrahy...)
Affinity DataEC50:  11.9nMAssay Description:Agonist activity at mu opioid receptor in Swiss albino mouse ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50318413(7alpha-(1-Hydroxy-1-methyl-ethyl)-6-ethoxy-6-demet...)
Affinity DataEC50:  44nMAssay Description:Agonist activity at mu opioid receptor in Swiss albino mouse ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50318412(7alpha-(1-Hydroxy-1-methyl-ethyl)-6-propoxy-6-deme...)
Affinity DataEC50:  1.99nMAssay Description:Agonist activity at mu opioid receptor in Swiss albino mouse ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50318415(7alpha-(1-Hydroxy-1-methyl-ethyl)-6-(cyclopropylme...)
Affinity DataEC50:  90nMAssay Description:Agonist activity at mu opioid receptor in Swiss albino mouse ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(MOUSE)
University Of Debrecen

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataEC50:  85.5nMAssay Description:Agonist activity at mu opioid receptor in Swiss albino mouse ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair