Affinity DataKi: 3.70E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 310nMAssay Description:Antagonist activity at human ERalpha expressed in human MCF7 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataIC50: 5.10E+3nMAssay Description:Antagonist activity at human ERalpha expressed in human MCF7 cells at 10 uM by luciferase reporter gene assayMore data for this Ligand-Target Pair