Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50039294
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50326694(5-Hydroxy-2-(4-hydroxyphenyl)-1-[4-(2-piperidin-1-...)
Affinity DataKi:  3.70E+3nMAssay Description:Displacement of [3H]CCPA from adenosine A1 receptor in rat brain cortical membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50326692(6-Hydroxy-2-phenyl-1-[4-(2-piperidin-1-ylethoxy)be...)
Affinity DataIC50:  310nMAssay Description:Antagonist activity at human ERalpha expressed in human MCF7 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50326693(2-(4-Hydroxyphenyl)-1-[4-(2-piperidin-1-ylethoxy)b...)
Affinity DataIC50:  5.10E+3nMAssay Description:Antagonist activity at human ERalpha expressed in human MCF7 cells at 10 uM by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed