Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 4819
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Mainz

LigandPNGBDBM82183((E)-[2-(dimethylamino)ethoxy]({[3-(2-fluoroethoxy)...)
Affinity DataKi:  57nM ΔG°:  -43.0kJ/molepH: 7.4 T: 2°CAssay Description:5-HT-2A receptor affinity was determined by a radioligand competition binding assay with GF-62 cells, a clonal cell line expressing high amounts of 5...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Mainz

LigandPNGBDBM82182(3-[2-(4-{[3-(2-fluoroethoxy)-2-methoxyphenyl](hydr...)
Affinity DataKi:  356nM ΔG°:  -38.3kJ/molepH: 7.4 T: 2°CAssay Description:5-HT-2A receptor affinity was determined by a radioligand competition binding assay with GF-62 cells, a clonal cell line expressing high amounts of 5...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Mainz

LigandPNGBDBM82181(3-(2-{4-[(2,3-dimethoxyphenyl)(hydroxy)methyl]pipe...)
Affinity DataKi:  390nM ΔG°:  -38.1kJ/molepH: 7.4 T: 2°CAssay Description:5-HT-2A receptor affinity was determined by a radioligand competition binding assay with GF-62 cells, a clonal cell line expressing high amounts of 5...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University Of Mainz

LigandPNGBDBM82184(3-(2-{4-[(2,3-dimethoxyphenyl)carbonyl]piperidin-1...)
Affinity DataKi:  411nM ΔG°:  -37.9kJ/molepH: 7.4 T: 2°CAssay Description:5-HT-2A receptor affinity was determined by a radioligand competition binding assay with GF-62 cells, a clonal cell line expressing high amounts of 5...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed