Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50032559
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50331020((S)-5-((2S,3S)-1-((2S,5S,8S,11S,20S)-8-((1H-imidaz...)
Affinity DataEC50:  1.12E+3nMAssay Description:Agonist activity at recombinant PTHR1 expressed in HEK293 cells co-transfected with CRE-Luc assessed as increase of adenylyl-cyclase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50331022((7S,10S,13S,16S,19S,22S,25S,28S)-13-((1H-imidazol-...)
Affinity DataEC50:  2.40nMAssay Description:Agonist activity at recombinant PTHR1 expressed in HEK293 cells co-transfected with CRE-Luc assessed as increase of adenylyl-cyclase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
University Of Padova

Curated by ChEMBL
LigandPNGBDBM50331021((S)-5-((2S,3S)-1-((3S,6S,9S,12S,15S)-6-((1H-imidaz...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at recombinant PTHR1 expressed in HEK293 cells co-transfected with CRE-Luc assessed as increase of adenylyl-cyclase activity after 4...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed