Compile Data Set for Download or QSAR
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Found 32 Enz. Inhib. hit(s) with all data for entry = 50032851
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50335620(2-(4-(4-(1H-indol-3-yl)piperidin-1-yl)butyl)-4-(2-...)
Affinity DataKi:  19.9nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50335618(2-{4-[4-(1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-y...)
Affinity DataKi:  28.3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301432(2-{4-[4-(1H-Indol-3-yl)-piperidin-1-yl]-butyl}-4-(...)
Affinity DataKi:  32.4nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301445(4-(2-Fluoro-phenyl)-2-{4-[4-(1H-indol-3-yl)-piperi...)
Affinity DataKi:  41.3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301428(2-{4-[4-(1H-Indol-3-yl)-piperidin-1-yl]-butyl}-4-p...)
Affinity DataKi:  42.4nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50335619(4-(4-chlorophenyl)-2-{4-[4-(1H-indol-3-yl)-3,6-dih...)
Affinity DataKi:  44.1nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301428(2-{4-[4-(1H-Indol-3-yl)-piperidin-1-yl]-butyl}-4-p...)
Affinity DataKi:  46.2nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50335621(4-(4-fluorophenyl)-2-{4-[4-(1H-indol-3-yl)-3,6-dih...)
Affinity DataKi:  47nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50335619(4-(4-chlorophenyl)-2-{4-[4-(1H-indol-3-yl)-3,6-dih...)
Affinity DataKi:  48.6nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301432(2-{4-[4-(1H-Indol-3-yl)-piperidin-1-yl]-butyl}-4-(...)
Affinity DataKi:  50.4nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301441(4-(2-Chloro-phenyl)-2-{4-[4-(1H-indol-3-yl)-piperi...)
Affinity DataKi:  62.3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50335621(4-(4-fluorophenyl)-2-{4-[4-(1H-indol-3-yl)-3,6-dih...)
Affinity DataKi:  62.3nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301445(4-(2-Fluoro-phenyl)-2-{4-[4-(1H-indol-3-yl)-piperi...)
Affinity DataKi:  68.4nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301444(2-{4-[4-(1H-Indol-3-yl)-piperidin-1-yl]-butyl}-4-o...)
Affinity DataKi:  69.1nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50335618(2-{4-[4-(1H-indol-3-yl)-3,6-dihydro-2H-pyridin-1-y...)
Affinity DataKi:  81.7nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301444(2-{4-[4-(1H-Indol-3-yl)-piperidin-1-yl]-butyl}-4-o...)
Affinity DataKi:  112nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301433(4-(4-Fluoro-phenyl)-2-{4-[4-(2-methyl-1H-indol-3-y...)
Affinity DataKi:  114nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50335620(2-(4-(4-(1H-indol-3-yl)piperidin-1-yl)butyl)-4-(2-...)
Affinity DataKi:  134nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301441(4-(2-Chloro-phenyl)-2-{4-[4-(1H-indol-3-yl)-piperi...)
Affinity DataKi:  147nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301433(4-(4-Fluoro-phenyl)-2-{4-[4-(2-methyl-1H-indol-3-y...)
Affinity DataKi:  147nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301436(4-(4-Methoxy-phenyl)-2-{4-[4-(2-methyl-1H-indol-3-...)
Affinity DataKi:  153nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301436(4-(4-Methoxy-phenyl)-2-{4-[4-(2-methyl-1H-indol-3-...)
Affinity DataKi:  184nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301437(2-{4-[4-(2-Methyl-1H-indol-3-yl)-piperidin-1-yl]-b...)
Affinity DataKi:  279nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301440(4-(2-Fluoro-phenyl)-2-{4-[4-(2-methyl-1H-indol-3-y...)
Affinity DataKi:  303nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301438(4-(2-Methoxy-phenyl)-2-{4-[4-(2-methyl-1H-indol-3-...)
Affinity DataKi:  319nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301434(4-(2-Chloro-phenyl)-2-{4-[4-(2-methyl-1H-indol-3-y...)
Affinity DataKi:  393nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 1A(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50335622(2-{4-[4-(2-methyl-1H-indol-3-yl)-3,6-dihydro-2H-py...)
Affinity DataKi:  642nMAssay Description:Displacement of [3H]8-OH-DPAT from 5-HT1A receptor in rat hippocampusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50335622(2-{4-[4-(2-methyl-1H-indol-3-yl)-3,6-dihydro-2H-py...)
Affinity DataKi:  882nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301440(4-(2-Fluoro-phenyl)-2-{4-[4-(2-methyl-1H-indol-3-y...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301438(4-(2-Methoxy-phenyl)-2-{4-[4-(2-methyl-1H-indol-3-...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301434(4-(2-Chloro-phenyl)-2-{4-[4-(2-methyl-1H-indol-3-y...)
Affinity DataKi:  1.30E+3nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Medical University Of Warsaw

Curated by ChEMBL
LigandPNGBDBM50301437(2-{4-[4-(2-Methyl-1H-indol-3-yl)-piperidin-1-yl]-b...)
Affinity DataKi:  1.80E+3nMAssay Description:Displacement of [3H]citalopram from SERT in rat cerebral cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed