Compile Data Set for Download or QSAR
maximum 50k data
Found 38 Enz. Inhib. hit(s) with all data for entry = 50033570
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347535(CHEMBL1801637)
Affinity DataIC50:  5nMAssay Description:Inhibition of human recombinant GSK3beta using prephosphorylated polypeptide substrate after 30 mins by Glow-type luminescence assay in presence of 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347531(CHEMBL1801633)
Affinity DataIC50:  47nMAssay Description:Inhibition of human recombinant GSK3beta using prephosphorylated polypeptide substrate after 30 mins by Glow-type luminescence assay in presence of 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM7876(2-bromo-1-(4-bromophenyl)ethan-1-one | Halomethyl ...)
Affinity DataIC50:  500nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347526(CHEMBL1801628)
Affinity DataIC50:  500nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347533(CHEMBL1801635)
Affinity DataIC50:  580nMAssay Description:Inhibition of human recombinant GSK3beta using prephosphorylated polypeptide substrate after 30 mins by Glow-type luminescence assay in presence of 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347534(CHEMBL1801636)
Affinity DataIC50:  890nMAssay Description:Inhibition of human recombinant GSK3beta using prephosphorylated polypeptide substrate after 30 mins by Glow-type luminescence assay in presence of 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347525(CHEMBL1801627)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM7879(2-bromo-1-(4-methoxyphenyl)ethan-1-one | CHEMBL103...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM7877(2-bromo-1-(4-chlorophenyl)ethan-1-one | Halomethyl...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347524(CHEMBL1801626)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347520(CHEMBL1801623)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347519(CHEMBL1801622)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347523(CHEMBL1801625)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50119691(2-Bromo-1-(4-nitro-phenyl)-ethanone | CHEMBL106072)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347527(CHEMBL1801629)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM7880(2-bromo-1-(4-phenylphenyl)ethan-1-one | CHEMBL4130...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM7878(2-bromo-1-(4-methylphenyl)ethan-1-one | Halomethyl...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM7874(2-chloro-1-(4-chlorophenyl)ethan-1-one | Halomethy...)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347508(CHEMBL1801611)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347530(CHEMBL1801632)
Affinity DataIC50:  4.47E+3nMAssay Description:Inhibition of human recombinant GSK3beta using prephosphorylated polypeptide substrate after 30 mins by Glow-type luminescence assay in presence of 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM7875(2-bromo-1-phenylethan-1-one | CHEMBL102953 | Halom...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347521(CHEMBL1800091)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50119685(2-Bromo-1-(4-trifluoromethyl-phenyl)-ethanone | CH...)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347522(CHEMBL1801624)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347513(CHEMBL1801616)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347532(CHEMBL1801634)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using prephosphorylated polypeptide substrate after 30 mins by Glow-type luminescence assay in presence of 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347511(CHEMBL1801614)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347529(CHEMBL1801631)
Affinity DataIC50:  1.34E+4nMAssay Description:Inhibition of human recombinant GSK3beta using prephosphorylated polypeptide substrate after 30 mins by Glow-type luminescence assay in presence of 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM7873(2-chloro-1-phenylethan-1-one | CHEMBL105712 | Halo...)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347528(CHEMBL1801630)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human recombinant GSK3beta using prephosphorylated polypeptide substrate after 30 mins by Glow-type luminescence assay in presence of 1...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347517(CHEMBL1801620)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347514(CHEMBL1801617)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347515(CHEMBL1801618)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347510(CHEMBL1801613)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347516(CHEMBL1801619)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347509(CHEMBL1801612)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347518(CHEMBL1801621)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Instituto De Qui£?Mica Medica-Csic

Curated by ChEMBL
LigandPNGBDBM50347512(CHEMBL1801615)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of GSK3beta using GS1 as substrate and [gamma-32P]ATP after 20 mins by radiometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed