Compile Data Set for Download or QSAR
maximum 50k data
Found 22 Enz. Inhib. hit(s) with all data for entry = 50033592
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50418829(CHEMBL1802381)
Affinity DataIC50:  10nMAssay Description:Inhibition of human Cdk1/cyclinB using histone H1 as a substrate and [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347865(CHEMBL1802383)
Affinity DataIC50:  20nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347864(CHEMBL1802382)
Affinity DataIC50:  60nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347868(CHEMBL1802387)
Affinity DataIC50:  90nMAssay Description:Inhibition of human Cdk1/cyclinB using histone H1 as a substrate and [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347866(CHEMBL1802384)
Affinity DataIC50:  130nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347870(CHEMBL1802869)
Affinity DataIC50:  390nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347869(CHEMBL1802388)
Affinity DataIC50:  620nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347863(CHEMBL1802870)
Affinity DataIC50:  770nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347868(CHEMBL1802387)
Affinity DataIC50:  920nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347863(CHEMBL1802870)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of hemaggutinin epitope-tagged human Nek2 transfected tetracycline-induced in human HEK293 cells pre-incubated for 45 mins by immunoprecip...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347866(CHEMBL1802384)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of human Cdk1/cyclinB using histone H1 as a substrate and [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347860(CHEMBL1802386)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of human Cdk1/cyclinB using histone H1 as a substrate and [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347867(CHEMBL1802385)
Affinity DataIC50:  4.90E+3nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase PLK1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347863(CHEMBL1802870)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human Plk1 using dephosphorylated alpha-casein as a substrate and [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347863(CHEMBL1802870)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human Cdk1/cyclinB using histone H1 as a substrate and [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347861(CHEMBL1802871)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347867(CHEMBL1802385)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human Cdk1/cyclinB using histone H1 as a substrate and [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347862(CHEMBL1802872)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347861(CHEMBL1802871)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human Cdk1/cyclinB using histone H1 as a substrate and [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase/G2/mitotic-specific cyclin- 1(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347862(CHEMBL1802872)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human Cdk1/cyclinB using histone H1 as a substrate and [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase Nek2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50347860(CHEMBL1802386)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human Nek2 in using [gamma-32P] ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM4814(CHEMBL535 | N-[2-(diethylamino)ethyl]-5-[(Z)-(5-fl...)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to human Cdk2More data for this Ligand-Target Pair