Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 8200
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236526(2-Ethoxy-10-[(2-N,N-dimethylamino-2-methyl)ethyl]b...)
Affinity DataKi:  11.1nM ΔG°:  -47.2kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236524( 2-Methoxy-10-[(2-N,N-dimethylamino-2-methyl)ethyl...)
Affinity DataKi:  11.6nM ΔG°:  -47.1kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236533(2-Fluoro-10-(2-N,N-dimethylaminoethyl)isoindolo[2,...)
Affinity DataKi:  24.3nM ΔG°:  -45.2kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236521(2-Phenyl-10-(2-N,N-dimethylaminoethyl)benzo[d]isot...)
Affinity DataKi:  26.8nM ΔG°:  -45.0kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236525(2-Methoxy-10-[(2-N,N-dimethylamino-2-ethyl)ethyl]b...)
Affinity DataKi:  28.3nM ΔG°:  -44.8kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236539(2-Fluoro-7-chloro-10-(2-N,N-dimethylaminoethyl)iso...)
Affinity DataKi:  37.6nM ΔG°:  -44.1kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236538(2-Methylthio-10-(2-N,N-dimethylaminoethyl)isoindol...)
Affinity DataKi:  49.7nM ΔG°:  -43.4kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236522(2-Bromo-10-[(2-N,N-dimethylamino-2-methyl)ethyl]be...)
Affinity DataKi:  54.1nM ΔG°:  -43.1kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236530(2-Isopropoxy-10-[(2-N,N-dimethylamino-2-methyl)eth...)
Affinity DataKi:  73.2nM ΔG°:  -42.4kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236534(2-Chloro-10-(2-N,N-dimethylaminoethyl)isoindolo[2,...)
Affinity DataKi:  80.7nM ΔG°:  -42.1kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236540(2-Phenyl-10-(2-N,N-dimethylaminoethyl)isoindolo[2,...)
Affinity DataKi:  84.6nM ΔG°:  -42.0kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236531(2-Methoxy-10-(2-N,N-dimethylaminoethyl)isoindolo[2...)
Affinity DataKi:  86.7nM ΔG°:  -41.9kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236520(10-[(2-N,N-Dimethylamino-2-methyl)ethyl]benzo[d]is...)
Affinity DataKi:  87.6nM ΔG°:  -41.9kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236537(10-(2-N,N-dimethylaminoethyl)benzo[d]isoindolo[2,1...)
Affinity DataKi:  92.6nM ΔG°:  -41.8kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236523(2-Methoxy-10-(2-N,N-dimethylaminoethyl)benzo[d]iso...)
Affinity DataKi:  96nM ΔG°:  -41.7kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236527(2-Benzyloxy-10-[(2-N,N-dimethylamino-2-methyl)ethy...)
Affinity DataKi:  100nM ΔG°:  -41.6kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236535(1-Chloro-10-(2-N,N-dimethylaminoethyl)-4-methyliso...)
Affinity DataKi:  104nM ΔG°:  -41.5kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236517(10-[(2-N,N-Dimethylamino-2-methyl)ethyl]-2-fluorob...)
Affinity DataKi:  116nM ΔG°:  -41.2kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236519(4-Chloro-10-(2-N,N-dimethylaminoethyl)benzo[d]isot...)
Affinity DataKi:  126nM ΔG°:  -41.0kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236543(10-(2-N,N-dimethylaminoethyl)isoindolo[2,1-a]indol...)
Affinity DataKi:  135nM ΔG°:  -40.8kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236536(2,4-Difluoro-10-(2-N,N-dimethylaminoethyl)isoindol...)
Affinity DataKi:  153nM ΔG°:  -40.5kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236544(2-Methoxy-10-[(2-N,N-dimethylamino-2-methyl)ethyl]...)
Affinity DataKi:  197nM ΔG°:  -39.8kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236528(2-Isopropoxy-10-[(2-N,N-dimethylamino-2-methyl)eth...)
Affinity DataKi:  239nM ΔG°:  -39.3kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236515(10-(2-N,N-Dimethylaminoethyl)benzo[d]isothiazolo[3...)
Affinity DataKi:  246nM ΔG°:  -39.2kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236516(10-(2-N,N-Dimethylaminoethyl)-2-fluorobenzo[d]isot...)
Affinity DataKi:  267nM ΔG°:  -39.0kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236518(10-(2-N,N-Dimethylaminoethyl)-2-methyl-8-methoxybe...)
Affinity DataKi:  269nM ΔG°:  -39.0kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236532(2-Methoxy-10-[(2-N,N-dimethylamino-2-methyl)ethyl]...)
Affinity DataKi:  279nM ΔG°:  -38.9kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236541(10-[(2-N,N-Dimethylamino-2-methyl)ethyl]isoindolo[...)
Affinity DataKi:  296nM ΔG°:  -38.8kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236542(2-Chloro-10-(2-N,N-dimethylaminoethyl)isoindolo[2,...)
Affinity DataKi:  393nM ΔG°:  -38.0kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Suven Life Sciences

LigandPNGBDBM236529(2-Cyclohexylmethyloxy-10-[(2-N,N-dimethylamino-2-m...)
Affinity DataKi: >1.00E+3nM ΔG°: >-35.6kJ/molepH: 7.4 T: 2°CAssay Description:In brief, receptor source and radioligand used were human recombinant expressed in HEK-293 cells and [3H] LSD (60-80 Ci/mmol), respectively. The fina...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed