Affinity DataIC50: 14nMAssay Description:Inhibition of CYP2D6 using dextromethorphan as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 189nMAssay Description:Inhibition of mouse Sky kinase assessed as inhibition of src substrate phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 246nMAssay Description:Inhibition of mouse Sky kinase assessed as inhibition of src substrate phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 476nMAssay Description:Inhibition of mouse Sky kinase assessed as inhibition of src substrate phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 495nMAssay Description:Inhibition of mouse Sky kinase assessed as inhibition of src substrate phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 501nMAssay Description:Inhibition of mouse Sky kinase assessed as inhibition of src substrate phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 560nMAssay Description:Inhibition of mouse Sky kinase assessed as inhibition of src substrate phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 598nMAssay Description:Inhibition of mouse Sky kinase assessed as inhibition of src substrate phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 655nMAssay Description:Inhibition of CYP2D6 using dextromethorphan as substrateMore data for this Ligand-Target Pair
Affinity DataIC50: 811nMAssay Description:Inhibition of mouse Sky kinase assessed as inhibition of src substrate phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 843nMAssay Description:Inhibition of mouse Sky kinase assessed as inhibition of src substrate phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of mouse Sky kinase assessed as inhibition of src substrate phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.13E+3nMAssay Description:Inhibition of mouse Sky kinase assessed as inhibition of src substrate phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.73E+3nMAssay Description:Inhibition of CK1deltaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.81E+3nMAssay Description:Inhibition of mouse Sky kinase assessed as inhibition of src substrate phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 2.20E+3nMAssay Description:Inhibition of mouse Sky kinase assessed as inhibition of src substrate phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 2.34E+3nMAssay Description:Inhibition of MerMore data for this Ligand-Target Pair
Affinity DataIC50: 2.44E+3nMAssay Description:Inhibition of MerMore data for this Ligand-Target Pair
Affinity DataIC50: 2.88E+3nMAssay Description:Inhibition of mouse Sky kinase assessed as inhibition of src substrate phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 4.41E+3nMAssay Description:Inhibition of mouse Sky kinase assessed as inhibition of src substrate phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 4.93E+3nMAssay Description:Inhibition of mouse Sky kinase assessed as inhibition of src substrate phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 5.25E+3nMAssay Description:Inhibition of AxlMore data for this Ligand-Target Pair
Affinity DataIC50: 6.61E+3nMAssay Description:Inhibition of CK1deltaMore data for this Ligand-Target Pair
Affinity DataIC50: 6.93E+3nMAssay Description:Inhibition of MerMore data for this Ligand-Target Pair
Affinity DataIC50: 8.66E+3nMAssay Description:Inhibition of mouse Sky kinase assessed as inhibition of src substrate phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of CK1deltaMore data for this Ligand-Target Pair
Affinity DataIC50: 1.84E+4nMAssay Description:Inhibition of AxlMore data for this Ligand-Target Pair
Affinity DataIC50: 1.94E+4nMAssay Description:Inhibition of AxlMore data for this Ligand-Target Pair
Affinity DataIC50: 2.19E+4nMAssay Description:Inhibition of VEGFR2More data for this Ligand-Target Pair
Affinity DataIC50: 2.27E+4nMAssay Description:Inhibition of FGFR1More data for this Ligand-Target Pair
Affinity DataIC50: 2.38E+4nMAssay Description:Inhibition of AxlMore data for this Ligand-Target Pair
Affinity DataIC50: 2.79E+4nMAssay Description:Inhibition of mouse Sky kinase assessed as inhibition of src substrate phosphorylation by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Chk1More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of INSRMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Chk1More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Chk1More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Chk1More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of AblMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of PKCzetaMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Cdk2More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Chk2More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Gsk3betaMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit beta(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of IKK-betaMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of IKKiMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of MAPKAP-2More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Pak4More data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Pfizer
Curated by ChEMBL
Pfizer
Curated by ChEMBL
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of PDK1More data for this Ligand-Target Pair
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of Pim-2More data for this Ligand-Target Pair