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Found 18 Enz. Inhib. hit(s) with all data for entry = 50034654
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50:  400nMAssay Description:Inhibition of rat DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50:  400nMAssay Description:Inhibition of rat DATMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50:  600nMAssay Description:Inhibition of rat DAT-mediated uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50:  600nMAssay Description:Inhibition of rat DAT-mediated uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of rat NET-mediated uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransporter(Rattus norvegicus (rat))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of rat NET-mediated uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50:  1.39E+5nMAssay Description:Inhibition of CYP3A4 in human microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A5(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50:  1.39E+5nMAssay Description:Inhibition of CYP3A5 in human microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A5(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50:  1.39E+5nMAssay Description:Inhibition of CYP3A5 in human microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50:  1.39E+5nMAssay Description:Inhibition of CYP3A4 in human microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50:  1.74E+5nMAssay Description:Inhibition of CYP2C19 in human microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C19(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50:  1.74E+5nMAssay Description:Inhibition of CYP2C19 in human microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50:  1.77E+5nMAssay Description:Inhibition of CYP2D6 in human microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2D6(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50:  1.77E+5nMAssay Description:Inhibition of CYP2D6 in human microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50:  2.33E+5nMAssay Description:Inhibition of CYP2C9 in human microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50:  2.33E+5nMAssay Description:Inhibition of CYP2C9 in human microsomeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of rat SERT-mediated uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Cephalon

Curated by ChEMBL
LigandPNGBDBM50365396(CHEMBL1956397)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of rat SERT-mediated uptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed