Found 26 Enz. Inhib. hit(s) with all data for entry = 50039612 
Affinity DataKi: 0.0490nMAssay Description:Displacement of [3H]DAMGO from mouse brain mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.0970nMAssay Description:Displacement of [3H]DAMGO from mouse brain mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 0.190nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.230nMAssay Description:Binding affinity to kappa opioid receptorMore data for this Ligand-Target Pair
3D Structure (crystal)
Affinity DataKi: 0.270nMAssay Description:Displacement of [3H]DAMGO from mouse brain mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Displacement of [3H]DAMGO from mouse brain mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Displacement of [3H]DAMGO from mouse brain mu opioid receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 0.290nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 0.340nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 0.350nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.410nMAssay Description:Displacement of [3H]DAMGO from mouse brain mu opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.450nMAssay Description:Displacement of [3H]DAMGO from mouse brain mu opioid receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 0.470nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.740nMAssay Description:Displacement of [3H]U-69,593 from mouse brain delta opioid receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 0.860nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.900nMAssay Description:Displacement of [3H]DAMGO from mouse brain mu opioid receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 1.42nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.28nMAssay Description:Displacement of [3H]U-69,593 from mouse brain delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.49nMAssay Description:Displacement of [3H]U-69,593 from mouse brain delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.12nMAssay Description:Displacement of [3H]U-69,593 from mouse brain delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 9.39nMAssay Description:Displacement of [3H]U-69,593 from mouse brain delta opioid receptorMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
Kitasato University
Curated by ChEMBL
Kitasato University
Curated by ChEMBL
Affinity DataKi: 9.91nMAssay Description:Displacement of [3H]DPDPE from kappa opioid receptor in guinea pig cerebellum membraneMore data for this Ligand-Target Pair
Affinity DataKi: 10.1nMAssay Description:Displacement of [3H]U-69,593 from mouse brain delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 12.1nMAssay Description:Displacement of [3H]U-69,593 from mouse brain delta opioid receptorMore data for this Ligand-Target Pair
Affinity DataKi: 13.5nMAssay Description:Displacement of [3H]U-69,593 from mouse brain delta opioid receptorMore data for this Ligand-Target Pair
