Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50039842
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50384998(CVD-0019905 | XANTHOHUMOL)
Affinity DataIC50:  6.60E+3nMAssay Description:Inhibition of human PDK1 assessed as inhibition of [33P] incorporation into substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50252521(CHEMBL492828 | isoxanthohumol)
Affinity DataIC50:  3.16E+4nMAssay Description:Inhibition of human PKC theta assessed as inhibition of [33P] incorporation into substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50252521(CHEMBL492828 | isoxanthohumol)
Affinity DataIC50:  4.53E+4nMAssay Description:Inhibition of human PKC alpha assessed as inhibition of [33P] incorporation into substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50252521(CHEMBL492828 | isoxanthohumol)
Affinity DataIC50:  5.87E+4nMAssay Description:Inhibition of human PDK1 assessed as inhibition of [33P] incorporation into substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C theta type(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50384998(CVD-0019905 | XANTHOHUMOL)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human PKC theta assessed as inhibition of [33P] incorporation into substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50384998(CVD-0019905 | XANTHOHUMOL)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human PKC alpha assessed as inhibition of [33P] incorporation into substrate after 60 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed