Compile Data Set for Download or QSAR
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Found 6 Enz. Inhib. hit(s) with all data for entry = 50004661
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50485345(CHEMBL2046656)
Affinity DataIC50:  1.30E+3nMAssay Description:Inhibition of partially purified human recombinant FTase measured for 15 mins by automated fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50485343(CHEMBL2046655)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of partially purified human recombinant FTase measured for 15 mins by automated fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50485344(CHEMBL2046654)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of partially purified human recombinant FTase measured for 15 mins by automated fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50485342(CHEMBL2046652)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of partially purified human recombinant FTase measured for 15 mins by automated fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50485346(CHEMBL2046653)
Affinity DataIC50:  8.30E+3nMAssay Description:Inhibition of partially purified human recombinant FTase measured for 15 mins by automated fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Homo sapiens (Human))
Al. I. Cuza University Of Iasi

Curated by ChEMBL
LigandPNGBDBM50485341(CHEMBL2046657)
Affinity DataIC50:  2.43E+4nMAssay Description:Inhibition of partially purified human recombinant FTase measured for 15 mins by automated fluorescence based assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed