Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50040508
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50395258(CHEMBL2163602)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of P300 CH1 domain-mediated HIF1 transcriptional activity in human LN229-V6R cells assessed as reduction in luciferase activity incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50395261(CHEMBL2163594)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of P300 CH1 domain-mediated HIF1 transcriptional activity in human LN229-V6R cells assessed as reduction in luciferase activity incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50395260(CHEMBL2163598)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of P300 CH1 domain-mediated HIF1 transcriptional activity in human LN229-V6R cells assessed as reduction in luciferase activity incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Emory University

Curated by ChEMBL
LigandPNGBDBM50395259(CHEMBL2163601)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of P300 CH1 domain-mediated HIF1 transcriptional activity in human LN229-V6R cells assessed as reduction in luciferase activity incubated ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed