Affinity DataKi: 1.90nMAssay Description:Binding affinity at endothelin receptor subtype AMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataKi: 10nMAssay Description:Binding affinity at type 1 angiotensin 2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 8.5nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.90nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.10nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 9.30nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.60nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.80nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 9.80nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.80nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 9.90nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 10.5nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
TargetType-1 angiotensin II receptor(Homo sapiens (Human))
China Pharmaceutical University
Curated by ChEMBL
China Pharmaceutical University
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Antagonist activity at type 1 angiotensin 2 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Antagonist activity at endothelin receptor subtype AMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 39nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 75nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 92nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 95nMAssay Description:Displacement of [125I]AngII from type 1 angiotensin 2 receptor in bovine adrenal cortexMore data for this Ligand-Target Pair
Affinity DataIC50: 99nMAssay Description:Antagonist activity at human endothelin receptor subtype A expressed in CHO-K1 cellsMore data for this Ligand-Target Pair