Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50004680
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of California Davis

Curated by ChEMBL
LigandPNGBDBM50485504(CHEMBL2069572)
Affinity DataEC50:  140nMAssay Description:Corrector activity at human CFTR deltaF508 mutant expressed in FRT cells stimulated forskolin and potentiator genistein with assessed as iodide influ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of California Davis

Curated by ChEMBL
LigandPNGBDBM50485505(CHEMBL2069648)
Affinity DataEC50:  1.60E+3nMAssay Description:Corrector activity at human CFTR deltaF508 mutant expressed in FRT cells stimulated forskolin and potentiator genistein with assessed as iodide influ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of California Davis

Curated by ChEMBL
LigandPNGBDBM50485508(CHEMBL2069571)
Affinity DataEC50:  4.90E+3nMAssay Description:Corrector activity at human CFTR deltaF508 mutant expressed in FRT cells stimulated forskolin and potentiator genistein with assessed as iodide influ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of California Davis

Curated by ChEMBL
LigandPNGBDBM50485507(CHEMBL2069570)
Affinity DataEC50:  1.50E+3nMAssay Description:Corrector activity at human CFTR deltaF508 mutant expressed in FRT cells stimulated forskolin and potentiator genistein with assessed as iodide influ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCystic fibrosis transmembrane conductance regulator(Homo sapiens (Human))
University Of California Davis

Curated by ChEMBL
LigandPNGBDBM50485506(CHEMBL2069649)
Affinity DataEC50:  4.60E+3nMAssay Description:Corrector activity at human CFTR deltaF508 mutant expressed in FRT cells stimulated forskolin and potentiator genistein with assessed as iodide influ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed