Compile Data Set for Download or QSAR
maximum 50k data
Found 30 Enz. Inhib. hit(s) with all data for entry = 50040725
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398987(CHEMBL2179712)
Affinity DataEC50:  2.90E+3nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50399002(CHEMBL2180076)
Affinity DataEC50:  468nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398989(CHEMBL2179710)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398990(CHEMBL2179709)
Affinity DataEC50:  680nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398991(CHEMBL2179708)
Affinity DataEC50:  1.50E+4nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398992(CHEMBL2180086)
Affinity DataEC50:  7.20E+3nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398993(CHEMBL2180085)
Affinity DataEC50:  660nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398994(CHEMBL2180084)
Affinity DataEC50:  260nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398995(CHEMBL2180083)
Affinity DataEC50:  560nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398996(CHEMBL2180082)
Affinity DataEC50:  5.40E+3nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398997(CHEMBL2180081)
Affinity DataEC50:  1.90E+4nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398998(CHEMBL2180080)
Affinity DataEC50:  1.90E+4nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398999(CHEMBL2180079)
Affinity DataEC50:  3.60E+3nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50399000(CHEMBL2180078)
Affinity DataEC50:  3.60E+4nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50399001(CHEMBL2180077)
Affinity DataEC50:  780nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50399002(CHEMBL2180076)
Affinity DataEC50:  470nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398987(CHEMBL2179712)
Affinity DataEC50:  2.88E+3nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398990(CHEMBL2179709)
Affinity DataEC50:  676nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398991(CHEMBL2179708)
Affinity DataEC50:  1.48E+4nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398992(CHEMBL2180086)
Affinity DataEC50:  7.24E+3nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398993(CHEMBL2180085)
Affinity DataEC50:  661nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398994(CHEMBL2180084)
Affinity DataEC50:  257nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398995(CHEMBL2180083)
Affinity DataEC50:  562nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398996(CHEMBL2180082)
Affinity DataEC50:  5.37E+3nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398997(CHEMBL2180081)
Affinity DataEC50:  1.95E+4nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398998(CHEMBL2180080)
Affinity DataEC50:  1.86E+4nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398999(CHEMBL2180079)
Affinity DataEC50:  3.55E+3nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50399000(CHEMBL2180078)
Affinity DataEC50:  3.63E+4nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50399001(CHEMBL2180077)
Affinity DataEC50:  776nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
University Of Troms£

Curated by ChEMBL
LigandPNGBDBM50398988(CHEMBL2179711)
Affinity DataEC50: >1.00E+5nMAssay Description:Antagonist activity against human CXCR4 expressed in COS7 cells assessed as inhibition of CXCL12-induced myo-[3H]inositol production by scintillation...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed