Affinity DataIC50: 2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 6nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 7nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 9nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 10nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))
Mrc Technology
Curated by ChEMBL
Mrc Technology
Curated by ChEMBL
Affinity DataIC50: 13nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
TargetMAP/microtubule affinity-regulating kinase 3(Homo sapiens (Human))
Mrc Technology
Curated by ChEMBL
Mrc Technology
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Mrc Technology
Curated by ChEMBL
Mrc Technology
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Inhibition of PDK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Mrc Technology
Curated by ChEMBL
Mrc Technology
Curated by ChEMBL
Affinity DataIC50: 30nMAssay Description:Inhibition of IKKepsilonMore data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Inhibition of TBK1-mediated RANTES release in LPS-stimulated mouse RAW264.7 cells compound incubated for 30 mins prior LPS challenge measured after 6...More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Mrc Technology
Curated by ChEMBL
Mrc Technology
Curated by ChEMBL
Affinity DataIC50: 68nMAssay Description:Inhibition of PDK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 81nMAssay Description:Inhibition of TBK1-mediated RANTES release in LPS-stimulated mouse RAW264.7 cells compound incubated for 30 mins prior LPS challenge measured after 6...More data for this Ligand-Target Pair
Affinity DataIC50: 88nMAssay Description:Inhibition of TBK1-mediated RANTES release in LPS-stimulated mouse RAW264.7 cells compound incubated for 30 mins prior LPS challenge measured after 6...More data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of TBK1-mediated RANTES release in LPS-stimulated mouse RAW264.7 cells compound incubated for 30 mins prior LPS challenge measured after 6...More data for this Ligand-Target Pair
Affinity DataIC50: 93nMAssay Description:Inhibition of TBK1-mediated RANTES release in LPS-stimulated mouse RAW264.7 cells compound incubated for 30 mins prior LPS challenge measured after 6...More data for this Ligand-Target Pair
TargetInhibitor of nuclear factor kappa-B kinase subunit epsilon(Homo sapiens (Human))
Mrc Technology
Curated by ChEMBL
Mrc Technology
Curated by ChEMBL
Affinity DataIC50: 100nMAssay Description:Inhibition of IKKepsilonMore data for this Ligand-Target Pair
Affinity DataIC50: 110nMAssay Description:Inhibition of TBK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of TBK1-mediated RANTES release in LPS-stimulated mouse RAW264.7 cells compound incubated for 30 mins prior LPS challenge measured after 6...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
Mrc Technology
Curated by ChEMBL
Mrc Technology
Curated by ChEMBL
Affinity DataIC50: 130nMAssay Description:Inhibition of PDK1 by radiometryMore data for this Ligand-Target Pair
Affinity DataIC50: 140nMAssay Description:Inhibition of TBK1-mediated RANTES release in LPS-stimulated mouse RAW264.7 cells compound incubated for 30 mins prior LPS challenge measured after 6...More data for this Ligand-Target Pair
Affinity DataIC50: 150nMAssay Description:Inhibition of TBK1-mediated RANTES release in LPS-stimulated mouse RAW264.7 cells compound incubated for 30 mins prior LPS challenge measured after 6...More data for this Ligand-Target Pair
Affinity DataIC50: 170nMAssay Description:Inhibition of TBK1-mediated RANTES release in LPS-stimulated mouse RAW264.7 cells compound incubated for 30 mins prior LPS challenge measured after 6...More data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of Aurora BMore data for this Ligand-Target Pair