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Found 6 Enz. Inhib. hit(s) with all data for entry = 50005251
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50489369(CHEMBL1232930 | GRL-0519)
Affinity DataKi:  0.5nMAssay Description:Inhibition of HIV-1 wildtype protease using Abz-Thr-Ile-Nle-p-nitro-Phe-Gln-Arg-NH2 as substrate incubated for 5 mins prior to substrate addition mea...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHIV-1 protease(Human immunodeficiency virus)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50489369(CHEMBL1232930 | GRL-0519)
Affinity DataKi:  1.20nMAssay Description:Inhibition of HIV-1 protease R8Q mutant using Abz-Thr-Ile-Nle-p-nitro-Phe-Gln-Arg-NH2 as substrate incubated for 5 mins prior to substrate addition m...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHIV-1 protease(Human immunodeficiency virus)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50489369(CHEMBL1232930 | GRL-0519)
Affinity DataKi:  3.20nMAssay Description:Inhibition of HIV-1 protease V82A mutant using Abz-Thr-Ile-Nle-p-nitro-Phe-Gln-Arg-NH2 as substrate incubated for 5 mins prior to substrate addition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHIV-1 protease(Human immunodeficiency virus)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50489369(CHEMBL1232930 | GRL-0519)
Affinity DataKi:  3.5nMAssay Description:Inhibition of HIV-1 protease I54M mutant using Abz-Thr-Ile-Nle-p-nitro-Phe-Gln-Arg-NH2 as substrate incubated for 5 mins prior to substrate addition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHIV-1 protease(Human immunodeficiency virus)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50489369(CHEMBL1232930 | GRL-0519)
Affinity DataKi:  8.90nMAssay Description:Inhibition of HIV-1 protease D30N mutant using Abz-Thr-Ile-Nle-p-nitro-Phe-Gln-Arg-NH2 as substrate incubated for 5 mins prior to substrate addition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetHIV-1 protease(Human immunodeficiency virus)
Georgia State University

Curated by ChEMBL
LigandPNGBDBM50489369(CHEMBL1232930 | GRL-0519)
Affinity DataKi:  31nMAssay Description:Inhibition of HIV-1 protease I50V mutant using Abz-Thr-Ile-Nle-p-nitro-Phe-Gln-Arg-NH2 as substrate incubated for 5 mins prior to substrate addition ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB