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Found 20 Enz. Inhib. hit(s) with all data for entry = 50042958
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433783(CHEMBL2381721)
Affinity DataKi:  29nMAssay Description:Inhibition of VMAT2-mediated [3H]DA uptake in rat striatal synaptic vesicles by liquid scintillation spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433777(CHEMBL2381727)
Affinity DataKi:  45nMAssay Description:Inhibition of VMAT2-mediated [3H]DA uptake in rat striatal synaptic vesicles by liquid scintillation spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433779(CHEMBL2381725)
Affinity DataKi:  49nMAssay Description:Inhibition of VMAT2-mediated [3H]DA uptake in rat striatal synaptic vesicles by liquid scintillation spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433780(CHEMBL2381724)
Affinity DataKi:  160nMAssay Description:Inhibition of VMAT2-mediated [3H]DA uptake in rat striatal synaptic vesicles by liquid scintillation spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433778(CHEMBL2381726)
Affinity DataKi:  170nMAssay Description:Inhibition of VMAT2-mediated [3H]DA uptake in rat striatal synaptic vesicles by liquid scintillation spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433774(CHEMBL2381720)
Affinity DataKi:  200nMAssay Description:Inhibition of VMAT2-mediated [3H]DA uptake in rat striatal synaptic vesicles by liquid scintillation spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433776(CHEMBL2381728)
Affinity DataKi:  269nMAssay Description:Inhibition of VMAT2-mediated [3H]DA uptake in rat striatal synaptic vesicles by liquid scintillation spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433781(CHEMBL2381723)
Affinity DataKi:  270nMAssay Description:Inhibition of VMAT2-mediated [3H]DA uptake in rat striatal synaptic vesicles by liquid scintillation spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433782(CHEMBL2381722)
Affinity DataKi:  279nMAssay Description:Inhibition of VMAT2-mediated [3H]DA uptake in rat striatal synaptic vesicles by liquid scintillation spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433777(CHEMBL2381727)
Affinity DataKi:  560nMAssay Description:Displacement of [3H]DTBZ from VMAT2 in Sprague-Dawley rat synaptic vesicle membranes after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433780(CHEMBL2381724)
Affinity DataKi:  2.28E+3nMAssay Description:Displacement of [3H]DTBZ from VMAT2 in Sprague-Dawley rat synaptic vesicle membranes after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433781(CHEMBL2381723)
Affinity DataKi:  2.35E+3nMAssay Description:Displacement of [3H]DTBZ from VMAT2 in Sprague-Dawley rat synaptic vesicle membranes after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433775(CHEMBL2381719)
Affinity DataKi:  3.78E+3nMAssay Description:Inhibition of VMAT2-mediated [3H]DA uptake in rat striatal synaptic vesicles by liquid scintillation spectroscopic analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433779(CHEMBL2381725)
Affinity DataKi:  3.94E+3nMAssay Description:Displacement of [3H]DTBZ from VMAT2 in Sprague-Dawley rat synaptic vesicle membranes after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433774(CHEMBL2381720)
Affinity DataKi:  4.06E+3nMAssay Description:Displacement of [3H]DTBZ from VMAT2 in Sprague-Dawley rat synaptic vesicle membranes after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433782(CHEMBL2381722)
Affinity DataKi:  5.91E+3nMAssay Description:Displacement of [3H]DTBZ from VMAT2 in Sprague-Dawley rat synaptic vesicle membranes after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433778(CHEMBL2381726)
Affinity DataKi:  6.76E+3nMAssay Description:Displacement of [3H]DTBZ from VMAT2 in Sprague-Dawley rat synaptic vesicle membranes after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433783(CHEMBL2381721)
Affinity DataKi:  8.29E+3nMAssay Description:Displacement of [3H]DTBZ from VMAT2 in Sprague-Dawley rat synaptic vesicle membranes after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433776(CHEMBL2381728)
Affinity DataKi:  8.47E+3nMAssay Description:Displacement of [3H]DTBZ from VMAT2 in Sprague-Dawley rat synaptic vesicle membranes after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSynaptic vesicular amine transporter(Rattus norvegicus (Rat))
University Of Arkansas For Medical Sciences

Curated by ChEMBL
LigandPNGBDBM50433775(CHEMBL2381719)
Affinity DataKi: >1.00E+5nMAssay Description:Displacement of [3H]DTBZ from VMAT2 in Sprague-Dawley rat synaptic vesicle membranes after 30 mins by scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed