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Found 7 Enz. Inhib. hit(s) with all data for entry = 50035885
TargetSodium-dependent dopamine transporter(BOVINE)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366564(CHEMBL1790051 | CHEMBL83729 | WIN-35065-2)
Affinity DataIC50:  22nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(BOVINE)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50366564(CHEMBL1790051 | CHEMBL83729 | WIN-35065-2)
Affinity DataIC50:  22nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(BOVINE)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50015692(8-Methyl-3-(4-nitro-phenyl)-8-aza-bicyclo[3.2.1]oc...)
Affinity DataIC50:  137nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(BOVINE)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50015692(8-Methyl-3-(4-nitro-phenyl)-8-aza-bicyclo[3.2.1]oc...)
Affinity DataIC50:  137nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(BOVINE)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM22418(Cocaine | Cocaine (-) | methyl (1R,2R,3S,5S)-3-(be...)
Affinity DataIC50:  139nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(BOVINE)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50015695(3-(4-Amino-phenyl)-8-methyl-8-aza-bicyclo[3.2.1]oc...)
Affinity DataIC50:  192nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(BOVINE)
University Of Maryland

Curated by ChEMBL
LigandPNGBDBM50015694(3-(2,4-Dinitro-phenyl)-8-methyl-8-aza-bicyclo[3.2....)
Affinity DataIC50:  1.10E+4nMAssay Description:Competitive inhibition against [3H]cocaine binding to cocaine receptor in bovine striatal tissueMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed