Compile Data Set for Download or QSAR
maximum 50k data
Found 12 Enz. Inhib. hit(s) with all data for entry = 50043190
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50437206(CHEMBL2402737)
Affinity DataIC50:  6nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50434287(CHEMBL2386346)
Affinity DataIC50:  18nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50437209(CHEMBL2402734)
Affinity DataIC50:  20nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50437208(CHEMBL2402735)
Affinity DataIC50:  21nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50437210(CHEMBL2402733)
Affinity DataIC50:  22nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50437212(CHEMBL2402731)
Affinity DataIC50:  22nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50437211(CHEMBL2402732)
Affinity DataIC50:  23nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50437207(CHEMBL2402736)
Affinity DataIC50:  25nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50437213(CHEMBL2402730)
Affinity DataIC50:  42nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50437214(CHEMBL2402729)
Affinity DataIC50:  56nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50437215(CHEMBL2402574)
Affinity DataIC50:  74nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetE3 ubiquitin-protein ligase Mdm2(Homo sapiens (Human))
Roche Research Center

Curated by ChEMBL
LigandPNGBDBM50437216(CHEMBL2402573)
Affinity DataIC50:  196nMAssay Description:Binding affinity to GST-tagged MDM2 (unknown origin) assessed as inhibition of interaction with p53 after 1 hr by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed