TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 51nMAssay Description:Displacement of fluorescein-labeled 25-hydroxycholesterol from human RORgammat LBD (262-518) Escherichia coli BL21(DE3) after 6 hrs by fluorescence p...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 51nMAssay Description:Displacement of fluorescein-labeled 25-hydroxycholesterol from human RORgammat LBD (262-518) Escherichia coli BL21(DE3) after 6 hrs by fluorescence p...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in HEK293t cells co-expressing Gal4-DNA binding domainMore data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 800nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.50E+3nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.30E+3nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 4.00E+3nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetThyroid hormone receptor alpha(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Antagonist activity at TRalpha (unknown origin) expressed in HEK293t cellsMore data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 4.70E+3nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 6.60E+3nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetOxysterols receptor LXR-alpha(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Antagonist activity at LXRalpha (unknown origin) expressed in HEK293t cellsMore data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.28E+4nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetThyroid hormone receptor beta(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.30E+4nMAssay Description:Antagonist activity at TRbeta (unknown origin) expressed in HEK293t cellsMore data for this Ligand-Target Pair
TargetSteroid hormone receptor ERR1(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.40E+4nMAssay Description:Antagonist activity at ERRalpha (unknown origin) expressed in HEK293t cellsMore data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.57E+4nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.25E+4nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.44E+4nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.90E+4nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: 3.00E+4nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair
TargetNuclear receptor ROR-gamma(Homo sapiens (Human))
New York University School Of Medicine
Curated by ChEMBL
New York University School Of Medicine
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Antagonist activity at transactivation domain of RORgammat (unknown origin) expressed in Drosophila Schneider cells co-expressing Gal4-DNA binding do...More data for this Ligand-Target Pair