Compile Data Set for Download or QSAR
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Found 11 Enz. Inhib. hit(s) with all data for entry = 50043555
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50005111(CHEMBL3086656)
Affinity DataKi:  4.50E+3nMAssay Description:Competitive inhibition of human recombinant DPP4 using AP-pNA as substrate preincubated for 30 mins followed by substrate addition measured after 30 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50005109(CHEMBL3086660)
Affinity DataKi:  5.00E+3nMAssay Description:Competitive inhibition of human recombinant DPP4 using AP-pNA as substrate preincubated for 30 mins followed by substrate addition measured after 30 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50005107(CHEMBL3086661)
Affinity DataKi:  6.30E+3nMAssay Description:Competitive inhibition of human recombinant DPP4 using AP-pNA as substrate preincubated for 30 mins followed by substrate addition measured after 30 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50005112(CHEMBL3086658)
Affinity DataKi:  6.10E+4nMAssay Description:Competitive inhibition of human recombinant DPP4 using AP-pNA as substrate preincubated for 30 mins followed by substrate addition measured after 30 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50005110(CHEMBL3086657)
Affinity DataKi:  1.42E+5nMAssay Description:Competitive inhibition of human recombinant DPP4 using AP-pNA as substrate preincubated for 30 mins followed by substrate addition measured after 30 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50152769(CHEMBL410972 | GLP-1(7-36)-NH2 | GLP-17-(7-36) der...)
Affinity DataIC50:  1.5nMAssay Description:Displacement of [125I]-exendin (9 to 39) from human GLP-1R expressed in African green monkey COS7 cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50442918(CHEMBL3086851)
Affinity DataIC50:  7.60nMAssay Description:Displacement of [125I]-exendin (9 to 39) from human GLP-1R expressed in African green monkey COS7 cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50442919(CHEMBL3086852)
Affinity DataIC50:  36nMAssay Description:Displacement of [125I]-exendin (9 to 39) from human GLP-1R expressed in African green monkey COS7 cells by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50152769(CHEMBL410972 | GLP-1(7-36)-NH2 | GLP-17-(7-36) der...)
Affinity DataEC50:  0.350nMAssay Description:Agonist activity at human GLP-1R expressed in African green monkey COS7 cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50442918(CHEMBL3086851)
Affinity DataEC50:  0.170nMAssay Description:Agonist activity at human GLP-1R expressed in African green monkey COS7 cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Tufts University

Curated by ChEMBL
LigandPNGBDBM50442919(CHEMBL3086852)
Affinity DataEC50:  0.260nMAssay Description:Agonist activity at human GLP-1R expressed in African green monkey COS7 cells assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed