Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with all data for entry = 50001542
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50016388(5-(2-Dimethylamino-ethyl)-4-methyl-2-(3-nitro-phen...)
Affinity DataKi:  505nMAssay Description:Inhibition of [3H]-diltiazem binding to calcium channels of guinea pig myocardiumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Oryctolagus cuniculus)
TBA

Curated by ChEMBL
LigandPNGBDBM50016385(4-Methyl-2-(3-nitro-phenyl)-2,5-dihydro-benzo[b][1...)
Affinity DataIC50:  140nMAssay Description:Reduction in amplitude of calcium-dependent slow-response action potential by blocking voltage sensitive calcium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50016388(5-(2-Dimethylamino-ethyl)-4-methyl-2-(3-nitro-phen...)
Affinity DataKd:  488nMAssay Description:Inhibition of [3H]-nitrendipine binding to calcium channels of guinea pig myocardiumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVoltage-dependent L-type calcium channel subunit alpha-1C(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50016385(4-Methyl-2-(3-nitro-phenyl)-2,5-dihydro-benzo[b][1...)
Affinity DataKd:  360nMAssay Description:Inhibition of [3H]-nitrendipine binding to calcium channels of guinea pig myocardiumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed