Affinity DataIC50: <2nMAssay Description:Inhibition of human JAK2More data for this Ligand-Target Pair
Affinity DataIC50: 2.70nMAssay Description:Inhibition of human CK2alpha2More data for this Ligand-Target Pair
Affinity DataIC50: <3nMAssay Description:Inhibition of Jak2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Inhibition of Jak2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: <3nMAssay Description:Inhibition of Jak2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: <3nMAssay Description:Inhibition of Jak2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: <3nMAssay Description:Inhibition of Jak1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Inhibition of Jak2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of Jak2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Inhibition of Jak2 in mouse BA/F3 cells expressing TEL-Jak2 assessed as inhibition of STAT5 phosphorylation by Western blotting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 15nMAssay Description:Inhibition of Jak2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Inhibition of Jak1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 22nMAssay Description:Inhibition of Jak1 (unknown origin)More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: 22nMAssay Description:Inhibition of human KDRMore data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of Jak2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 24nMAssay Description:Inhibition of Jak1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 25nMAssay Description:Inhibition of human AblMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of Jak2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of Jak2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Inhibition of Jak1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Inhibition of Jak1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition of human FgrMore data for this Ligand-Target Pair
Affinity DataIC50: 33nMAssay Description:Inhibition of Jak2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of human JAK3More data for this Ligand-Target Pair
Affinity DataIC50: 35nMAssay Description:Inhibition of human TrkAMore data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 3(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: 40nMAssay Description:Inhibition of human Flt4More data for this Ligand-Target Pair
Affinity DataIC50: 45nMAssay Description:Inhibition of human Flt3More data for this Ligand-Target Pair
TargetProto-oncogene tyrosine-protein kinase receptor Ret(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: 46nMAssay Description:Inhibition of human RetMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of human FGFR1More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of Jak2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Inhibition of human ALKMore data for this Ligand-Target Pair
Affinity DataIC50: 58nMAssay Description:Inhibition of human aurora A kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 63nMAssay Description:Inhibition of human LIMK1More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Inhibition of Jak2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 131nMAssay Description:Inhibition of Jak1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 190nMAssay Description:Inhibition of human SIKMore data for this Ligand-Target Pair
Affinity DataIC50: 200nMAssay Description:Inhibition of human PKCzetaMore data for this Ligand-Target Pair
Affinity DataIC50: 220nMAssay Description:Inhibition of Jak3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 240nMAssay Description:Inhibition of Tyk2 in mouse BA/F3 cells expressing TEL-Tyk2 assessed as inhibition of STAT5 phosphorylation by Western blotting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Inhibition of Jak1 in mouse BA/F3 cells expressing TEL-Jak1 assessed as inhibition of STAT5 phosphorylation by Western blotting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 490nMAssay Description:Inhibition of Jak2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 670nMAssay Description:Inhibition of Jak2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 800nMAssay Description:Inhibition of Jak2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.44E+3nMAssay Description:Inhibition of Jak3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of Jak1 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 1.82E+3nMAssay Description:Inhibition of Jak3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of Jak3 in mouse BA/F3 cells expressing TEL-Jak3 assessed as inhibition of STAT5 phosphorylation by Western blotting analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 2.46E+3nMAssay Description:Inhibition of Jak3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.78E+3nMAssay Description:Inhibition of Jak3 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 3.93E+3nMAssay Description:Inhibition of Jak3 (unknown origin)More data for this Ligand-Target Pair