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Found 37 Enz. Inhib. hit(s) with all data for entry = 50044629
TargetSodium-dependent dopamine transporter(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023181(CHEMBL3298876)
Affinity DataKi:  1.01E+3nMAssay Description:Inhibition of DAT (unknown origin)-mediated dopamine reuptakeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023162(CHEMBL3298862)
Affinity DataIC50:  294nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023163(CHEMBL3298863)
Affinity DataIC50:  369nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023165(CHEMBL3298865)
Affinity DataIC50:  386nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023161(CHEMBL3298870)
Affinity DataIC50:  425nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50302907(2-(N-Cyclopropylamino)-3-chloropropiophenone | CHE...)
Affinity DataIC50:  533nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023177(CHEMBL3298871)
Affinity DataIC50:  592nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50302937(2-(N-Propylamino)-3'-chloropropiophenone | CHEMBL5...)
Affinity DataIC50:  793nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023176(CHEMBL3298869)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023173(CHEMBL3298866)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023175(CHEMBL3298868)
Affinity DataIC50:  2.01E+3nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023174(CHEMBL3298867)
Affinity DataIC50:  2.37E+3nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50028642(1-Benzyl-butylamine | CHEMBL25435)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50302907(2-(N-Cyclopropylamino)-3-chloropropiophenone | CHE...)
Affinity DataIC50:  3.18E+3nMAssay Description:Inhibition of SERT-mediated serotonin uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023164(CHEMBL3298864)
Affinity DataIC50:  5.92E+3nMAssay Description:Inhibition of DAT-mediated dopamine uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50302937(2-(N-Propylamino)-3'-chloropropiophenone | CHEMBL5...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SERT-mediated serotonin uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50028642(1-Benzyl-butylamine | CHEMBL25435)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SERT-mediated serotonin uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023180(CHEMBL3298875)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SERT-mediated serotonin uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023164(CHEMBL3298864)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of SERT-mediated serotonin uptake in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Homo sapiens (Human))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023181(CHEMBL3298876)
Affinity DataEC50:  2.12E+3nMAssay Description:Induction of SERT (unknown origin)-mediated serotonin releaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023177(CHEMBL3298871)
Affinity DataEC50:  181nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50029103(2-(3-Chloro-phenyl)-1-methyl-ethylamine | CHEMBL14...)
Affinity DataEC50:  120nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023178(CHEMBL3298873)
Affinity DataEC50:  410nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023179(CHEMBL3298874)
Affinity DataEC50:  4.70E+3nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50302907(2-(N-Cyclopropylamino)-3-chloropropiophenone | CHE...)
Affinity DataEC50:  1.33E+3nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023162(CHEMBL3298862)
Affinity DataEC50:  562nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023163(CHEMBL3298863)
Affinity DataEC50:  733nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023165(CHEMBL3298865)
Affinity DataEC50:  621nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023173(CHEMBL3298866)
Affinity DataEC50:  1.07E+3nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023174(CHEMBL3298867)
Affinity DataEC50:  1.01E+3nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023175(CHEMBL3298868)
Affinity DataEC50:  1.63E+3nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023161(CHEMBL3298870)
Affinity DataEC50:  356nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent serotonin transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023176(CHEMBL3298869)
Affinity DataEC50:  667nMAssay Description:Induction of SERT-mediated serotonin release in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023180(CHEMBL3298875)
Affinity DataEC50:  411nMAssay Description:Induction of DAT-mediated dopamine release in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023179(CHEMBL3298874)
Affinity DataEC50:  225nMAssay Description:Induction of DAT-mediated dopamine release in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50029103(2-(3-Chloro-phenyl)-1-methyl-ethylamine | CHEMBL14...)
Affinity DataEC50:  12nMAssay Description:Induction of DAT-mediated dopamine release in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium-dependent dopamine transporter(Rattus norvegicus (rat))
Rti International

Curated by ChEMBL
LigandPNGBDBM50023178(CHEMBL3298873)
Affinity DataEC50:  47nMAssay Description:Induction of DAT-mediated dopamine release in rat synaptosomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed