Compile Data Set for Download or QSAR
maximum 50k data
Found 24 Enz. Inhib. hit(s) with all data for entry = 50035785
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50452590(CHEMBL3084309)
Affinity DataKi:  0.940nMAssay Description:The compound was tested for the ability to displace opioid receptor kappa specific radioligand [3H]DADLEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50001465((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataKi:  1.5nMAssay Description:The compound was tested for the ability to displace opioid receptor kappa specific radioligand [3H]DADLEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50016829(10-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-1...)
Affinity DataKi:  2.30nMAssay Description:The compound was tested for the ability to displace delta-receptor specific radioligand [3H]DSLETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50016829(10-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-1...)
Affinity DataKi:  2.30nMAssay Description:The compound was tested for the ability to displace opioid receptor delta specific radioligand [3H]-DSLETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50001465((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataKi:  2.5nMAssay Description:The compound was tested for the ability to displace delta-receptor specific radioligand [3H]DSLETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50452590(CHEMBL3084309)
Affinity DataKi:  3.30nMAssay Description:The compound was tested for the ability to displace delta-receptor specific radioligand [3H]DSLETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50016830(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi:  3.5nMAssay Description:The compound was tested for the ability to displace opioid receptor kappa specific radioligand [3H]DADLEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50016833(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi:  5.40nMAssay Description:The compound was tested for the ability to displace opioid receptor kappa specific radioligand [3H]DADLEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50016833(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi:  5.40nMAssay Description:The compound was tested for the ability to displace opioid receptor kappa specific radioligand [3H]DADLEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50001465((S)-2-[(S)-2-(2-{2-[(S)-2-Amino-3-(4-hydroxy-pheny...)
Affinity DataKi:  9.40nMAssay Description:The compound was tested for the ability to displace Opioid receptor mu 1 specific radioligand [3H]DAGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50016834(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi:  12nMAssay Description:The compound was tested for the ability to displace opioid receptor kappa specific radioligand [3H]naloxoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50452590(CHEMBL3084309)
Affinity DataKi:  14nMAssay Description:The compound was tested for the ability to displace Opioid receptor mu 1 specific radioligand [3H]DAGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50016832(19-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-1...)
Affinity DataKi:  15nMAssay Description:The compound was tested for the ability to displace receptor specific radioligand [3H]DPDPEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50016829(10-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-1...)
Affinity DataKi:  21nMAssay Description:The compound was tested for the ability to displace mu-receptor specific radioligand [3H]DAGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50016830(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi:  22nMAssay Description:The compound was tested for the ability to displace opioid receptor kappa specific radioligand [3H]naloxoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50452589(CHEMBL2370362)
Affinity DataKi:  26nMAssay Description:The compound was tested for the ability to displace opioid receptor kappa specific radioligand [3H]DADLEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50016832(19-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-1...)
Affinity DataKi:  31nMAssay Description:The compound was tested for the ability to displace opioid receptor delta specific radioligand [3H]-DSLETMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50452589(CHEMBL2370362)
Affinity DataKi:  157nMAssay Description:The compound was tested for the ability to displace opioid receptor kappa specific radioligand [3H]naloxoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50016834(13-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-7...)
Affinity DataKi:  178nMAssay Description:The compound was tested for the ability to displace opioid receptor kappa specific radioligand [3H]DADLEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50016832(19-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-1...)
Affinity DataKi:  387nMAssay Description:The compound was tested for the ability to displace delta-receptor specific radioligand [3H]DPDPEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50016832(19-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-1...)
Affinity DataKi:  683nMAssay Description:The compound was tested for the ability to displace delta-receptor specific radioligand [3H]DPDPEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50016832(19-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-1...)
Affinity DataKi:  1.80E+3nMAssay Description:The compound was tested for the ability to displace delta-receptor specific radioligand [3H]DPDPEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50016832(19-[2-Amino-3-(4-hydroxy-phenyl)-propionylamino]-1...)
Affinity DataKi:  1.80E+3nMAssay Description:The compound was tested for the ability to displace mu-receptor specific radioligand [3H]DAGOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Rattus norvegicus (rat))
Smith Kline And French Laboratories

Curated by ChEMBL
LigandPNGBDBM50228042(CHEMBL323548)
Affinity DataIC50:  0.0187nMAssay Description:The compound was tested for the ability to displace delta-receptor specific radioligand [3H]DPDPEMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed