BindingDB PrimarySearch

Found 21 Enz. Inhib. hit(s) with all data for entry = 50046181

D(3) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50071959(9H-Fluorene-2-carboxylic acid {4-[4-(2,3-dichloro-...)

Ki: 0.233nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway
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D(3) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50161214(CHEMBL180010 | N-(4-(4-(2,3-dichlorophenyl)piperaz...)

Ki: 0.316nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway
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D(2) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)

Ki: 0.343nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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D(3) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50378008(CHEMBL1627314)

Ki: 0.920nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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D(3) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)

Ki: 1nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway
UniProtKB/SwissProt
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D(3) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50097908(CHEMBL3590086)

Ki: 2.10nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor assessed as inhibition constant for lower affinity site expressed in HEK293 cel...More data for this Ligand-Target Pair

PDB Reactome pathway
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D(3) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50097908(CHEMBL3590086)

Ki: 3nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway
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D(3) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50097922(CHEMBL3590085)

Ki: 3.20nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway
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D(2) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50097908(CHEMBL3590086)

Ki: 47nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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D(2) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50071959(9H-Fluorene-2-carboxylic acid {4-[4-(2,3-dichloro-...)

Ki: 55nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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D(4) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50130293(7-{4-[4-(2,3-dichlorophenyl)piperazin-1-yl]butoxy}...)

Ki: 57nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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D(2) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50161214(CHEMBL180010 | N-(4-(4-(2,3-dichlorophenyl)piperaz...)

Ki: 74nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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D(2) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50378008(CHEMBL1627314)

Ki: 217nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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D(2) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50097908(CHEMBL3590086)

Ki: 335nMAssay Description:Binding affinity to human dopamine D2 receptorMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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D(4) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50161214(CHEMBL180010 | N-(4-(4-(2,3-dichlorophenyl)piperaz...)

Ki: 550nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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D(4) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50378008(CHEMBL1627314)

Ki: 2.04E+3nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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D(2) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50097922(CHEMBL3590085)

Ki: 2.11E+3nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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D(4) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50097908(CHEMBL3590086)

Ki: 2.37E+3nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

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D(4) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50071959(9H-Fluorene-2-carboxylic acid {4-[4-(2,3-dichloro-...)

Ki: 3.67E+3nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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DrugBank antibodypedia GoogleScholar

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D(4) dopamine receptor(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50097922(CHEMBL3590085)

Ki: 3.56E+4nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Potassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
National Institute On Drug Abuse-Intramural Research Program

Curated by ChEMBL

BDBM50342720((R)-N-(4-(4-(2,3-dichlorophenyl)piperazin-1-yl)-3-...)

IC50: 380nMAssay Description:Inhibition of human ERG by PatchXpress assayMore data for this Ligand-Target Pair

PDB MMDB Reactome pathway KEGG
UniProtKB/SwissProt UniProtKB/TrEMBL
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